SCHEMBL997429

SCHEMBL997429

CCSCC(Oc1ccc(Cl)cc1)N1CCCC1

nearest known ligand 0.39

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
TP53 P04637 2/20 0.39
LMNA P02545 1/20 0.38
KMT2A Q03164 1/20 0.38
SIGMAR1 Q99720 5/20 0.37
THRB P10828 1/20 0.37
LTA4H P09960 1/20 0.35
PTGS2 P35354 1/20 0.35
HRH3 Q9Y5N1 6/20 0.35
POLB P06746 1/20 0.35
MAPT P10636 1/20 0.35
HPGD P15428 1/20 0.35
RAB9A P51151 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL997427 1.00 TP53 (0.39) TP53LMNAKMT2ASIGMAR1THRB
SCHEMBL999194 0.85 SLC6A4 (0.43) HRH3POLB
SCHEMBL999196 0.85 SLC6A4 (0.43) HRH3POLB
SCHEMBL998852 0.82 SLC6A4 (0.41) TP53LMNAKMT2ASIGMAR1LTA4H
SCHEMBL998851 0.82 SLC6A4 (0.41) TP53LMNAKMT2ASIGMAR1LTA4H
SCHEMBL1002884 0.82 CYP1A2 (0.42) TP53LMNAKMT2APOLBMAPT
SCHEMBL1002885 0.82 CYP1A2 (0.42) TP53LMNAKMT2APOLBMAPT
SCHEMBL1002277 0.78 HTR7 (0.42) TP53LMNAKMT2ASIGMAR1LTA4H
SCHEMBL992649 0.78 HRH3 (0.40) TP53SIGMAR1HRH3
SCHEMBL1002275 0.78 HTR7 (0.42) TP53LMNAKMT2ASIGMAR1LTA4H

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2456436-A1 3-PHENOXYMETHYLPYRROLIDINE COMPOUNDS Theravance, Inc. (US) 2012-05-30 EP disclosed
WO-2011011231-A1 3-PHENOXYMETHYLPYRROLIDINE COMPOUNDS THERAVANCE, INC. (US) 2011-01-27 WO disclosed