SCHEMBL998852

SCHEMBL998852

CCSCC(Oc1ccc(C(F)(F)F)cc1)N1CCCC1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SLC6A4 P31645 7/20 0.41
LTA4H P09960 1/20 0.39
MC4R P32245 1/20 0.39
HRH3 Q9Y5N1 4/20 0.38
MMP2 P08253 1/20 0.36
MMP9 P14780 1/20 0.36
KDM4E B2RXH2 3/20 0.36
ALDH1A1 P00352 2/20 0.36
OPRK1 P41145 2/20 0.35
SLC6A2 P23975 3/20 0.34
SLC6A3 Q01959 3/20 0.34
NPC1 O15118 2/20 0.34
CYP2D6 P10635 2/20 0.34
CYP2C19 P33261 2/20 0.34
MTOR P42345 2/20 0.34
RAB9A P51151 2/20 0.34
KCNK2 O95069 2/20 0.34
KCNH2 Q12809 2/20 0.34
CACNA1C Q13936 2/20 0.34
MEN1 O00255 2/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL998851 1.00 SLC6A4 (0.41) SLC6A4LTA4HMC4RHRH3MMP2
SCHEMBL997429 0.82 TP53 (0.39) LTA4HHRH3RAB9AKMT2ALMNA
SCHEMBL997427 0.82 TP53 (0.39) LTA4HHRH3RAB9AKMT2ALMNA
SCHEMBL994992 0.80 SLC6A4 (0.48) SLC6A4LTA4HHRH3KDM4EALDH1A1
SCHEMBL996214 0.80 SLC6A4 (0.42) SLC6A4LTA4HHRH3MMP2MMP9
SCHEMBL996213 0.80 SLC6A4 (0.42) SLC6A4LTA4HHRH3MMP2MMP9
SCHEMBL14829991 0.76 MMP2 (0.45) SLC6A4LTA4HHRH3MMP2MMP9
SCHEMBL999194 0.76 SLC6A4 (0.43) SLC6A4HRH3KDM4EALDH1A1SLC6A2
SCHEMBL999196 0.76 SLC6A4 (0.43) SLC6A4HRH3KDM4EALDH1A1SLC6A2
SCHEMBL1079982 0.74 CYP2C8 (0.35) SLC6A4CYP2C9TSHRDRD2HTR2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2456436-A1 3-PHENOXYMETHYLPYRROLIDINE COMPOUNDS Theravance, Inc. (US) 2012-05-30 EP disclosed
WO-2011011231-A1 3-PHENOXYMETHYLPYRROLIDINE COMPOUNDS THERAVANCE, INC. (US) 2011-01-27 WO disclosed