SCHEMBL9975899

SCHEMBL9975899

COC(=O)c1sc(C2(C)CC2)cc1C1=C(C2CCC(C)CC2)CN(C)CC1

nearest known ligand 0.34

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
TP53 P04637 1/20 0.34
MAPT P10636 1/20 0.34
TLR2 O60603 1/20 0.32
ALDH1A1 P00352 3/20 0.31
TSHR P16473 1/20 0.31
OPRM1 P35372 1/20 0.30
KDM4E B2RXH2 1/20 0.30
KMT2A Q03164 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10381852 0.90 ADRA2C (0.31)
SCHEMBL19397895 0.85 ALDH1A1 (0.38) TP53MAPTTLR2ALDH1A1TSHR
SCHEMBL9975903 0.84 MAPT (0.36) TP53MAPTTLR2ALDH1A1TSHR
SCHEMBL10364454 0.83 TP53 (0.32) TP53MAPTTLR2
SCHEMBL10382630 0.82 RAF1 (0.41) TP53MAPTTLR2
SCHEMBL10364962 0.82 KDM4E (0.45) TP53MAPTALDH1A1KDM4EKMT2A
SCHEMBL9975909 0.80 SLC6A3 (0.37) TP53MAPTTLR2ALDH1A1KDM4E
SCHEMBL9975697 0.80 MAPT (0.39) TP53MAPTTLR2ALDH1A1KDM4E
SCHEMBL9975771 0.79 NR1I2 (0.40) TP53MAPTTLR2ALDH1A1TSHR
SCHEMBL9975732 0.78 ALDH1A1 (0.45) TP53MAPTALDH1A1TSHRKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012083105-A1 INHIBITORS OF HEPATITIS C VIRUS POLYMERASE COCRYSTAL DISCOVERY, INC. (US) 2012-06-21 WO disclosed