SCHEMBL997628

SCHEMBL997628

CC(=O)N1C(c2cccc(F)c2)c2[nH]c3nccnc3c2CC12CC2

nearest known ligand 0.37

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
KIF11 P52732 4/20 0.37
RXFP1 Q9HBX9 2/20 0.37
SLC40A1 Q9NP59 1/20 0.36
ALDH1A1 P00352 2/20 0.34
CYP2D6 P10635 1/20 0.34
TNKS O95271 4/20 0.33
TDP1 Q9NUW8 1/20 0.33
TP53 P04637 1/20 0.33
KDM4E B2RXH2 1/20 0.32
PKM P14618 1/20 0.32
HDAC4 P56524 1/20 0.32
HPGD P15428 1/20 0.32
HTT P42858 1/20 0.32
EP300 Q09472 1/20 0.32
CREBBP Q92793 1/20 0.32
OPRK1 P41145 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL999387 0.91 KIF11 (0.36) KIF11RXFP1SLC40A1ALDH1A1CYP2D6
SCHEMBL999103 0.88 KIF11 (0.40) KIF11RXFP1SLC40A1CYP2D6TNKS
SCHEMBL998439 0.86 KIF11 (0.37) KIF11SLC40A1ALDH1A1CYP2D6TP53
SCHEMBL999207 0.82 KIF11 (0.38) KIF11RXFP1ALDH1A1CYP2D6
SCHEMBL997542 0.82 KIF11 (0.38) KIF11RXFP1SLC40A1ALDH1A1TDP1
SCHEMBL998181 0.81 KIF11 (0.42) KIF11RXFP1ALDH1A1TDP1TP53
SCHEMBL998701 0.80 KIF11 (0.50) KIF11TDP1TP53KDM4E
SCHEMBL998800 0.80 KIF11 (0.39) KIF11RXFP1SLC40A1ALDH1A1CYP2D6
SCHEMBL1000704 0.79 KIF11 (0.36) KIF11RXFP1SLC40A1ALDH1A1CYP2D6
SCHEMBL996597 0.76 KIF11 (0.39) KIF11RXFP1SLC40A1ALDH1A1CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7872133-B2 Tricyclic heterocycle compound ONO PHARMACEUTICAL CO., LTD. (JP) 2011-01-18 US disclosed