SCHEMBL997654

SCHEMBL997654

CCOC(=O)N(CC)c1cccc2c(N(CC)C(=O)OCC)cccc12

nearest known ligand 0.43

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 2/20 0.43
GAA P10253 1/20 0.43
TSHR P16473 4/20 0.43
ALDH1A1 P00352 4/20 0.41
KDM4E B2RXH2 1/20 0.41
CA12 O43570 1/20 0.41
CA1 P00915 1/20 0.41
CA2 P00918 1/20 0.41
CA7 P43166 1/20 0.41
CA9 Q16790 1/20 0.41
CA14 Q9ULX7 1/20 0.41
CDC25B P30305 3/20 0.40
LMNA P02545 2/20 0.40
NPSR1 Q6W5P4 1/20 0.40
CYP3A4 P08684 2/20 0.40
HPGD P15428 1/20 0.40
CYP1A2 P05177 1/20 0.40
CDC25A P30304 1/20 0.39
CDC25C P30307 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8966581 0.91 SIGMAR1 (0.56) SIGMAR1TSHRALDH1A1KDM4ECDC25B
SCHEMBL996368 0.84 ALDH1A1 (0.45) GAAALDH1A1CA12CA1CA2
SCHEMBL995336 0.81 CA12 (0.46) SIGMAR1GAATSHRALDH1A1CA12
SCHEMBL18249419 0.79 KDM4E (0.48) GAATSHRALDH1A1KDM4ECA12
SCHEMBL9224528 0.77 TSHR (0.50) TSHRALDH1A1CA12CA1CA2
SCHEMBL20164248 0.76 PTGS2 (0.42) TSHRALDH1A1KDM4ELMNACYP3A4
SCHEMBL15016098 0.75 HPGD (0.41) GAATSHRALDH1A1KDM4ECDC25B
SCHEMBL27466253 0.75 TSHR (0.47) TSHRALDH1A1CDC25BLMNACYP3A4
SCHEMBL798942 0.75 NR4A2 (0.49) ALDH1A1LMNANPSR1CYP3A4CYP1A2
SCHEMBL18249478 0.75 TSHR (0.41) TSHRALDH1A1KDM4ELMNANPSR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8809574-B2 Method for preparing isocyanates by liquid-phase thermal cracking LANZHOU INSTITUTE OF CHEMICAL PHYSICS, CHINESE ACADEMY OF SCIENCES (CN) 2014-08-19 US disclosed
US-20110021810-A1 METHOD FOR PREPARING ISOCYANATES BY LIQUID-PHASE THERMAL CRACKING LANZHOU INSTITUTE OF CHEMICAL PHYSICS, CHINESE ACADEMY OF SCIENCES (CN) 2011-01-27 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20110021810-A1 METHOD FOR PREPARING ISOCYANATES BY LIQUID-PHASE THERMAL CRACKING DBI, CCNI, DGKI SIGMAR1 1697/4885GAA 4550/4885TSHR 4586/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.