SCHEMBL997714

SCHEMBL997714

N#CC(O)(c1ccccc1)C(F)(F)F

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.42
TSHR P16473 1/20 0.42
PTPN1 P18031 1/20 0.39
NR1H2 P55055 5/20 0.37
NR1H3 Q13133 3/20 0.36
ATM Q13315 1/20 0.36
CYP2D6 P10635 2/20 0.35
DRD2 P14416 1/20 0.35
DRD4 P21917 1/20 0.35
OPRM1 P35372 1/20 0.35
DRD3 P35462 1/20 0.35
CYP1A2 P05177 1/20 0.34
CYP2C9 P11712 1/20 0.34
CYP2C19 P33261 1/20 0.34
AR P10275 1/20 0.34
CYP19A1 P11511 1/20 0.34
HSD11B1 P28845 2/20 0.33
S1PR4 O95977 1/20 0.33
LMNA P02545 1/20 0.33
MAPT P10636 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL611603 0.78 TSHR (0.42) ALDH1A1TSHRPTPN1NR1H2NR1H3
SCHEMBL14101146 0.78 TSHR (0.42) ALDH1A1TSHRPTPN1ATMCYP2D6
SCHEMBL16428437 0.77 TSHR (0.46) ALDH1A1TSHRPTPN1NR1H2NR1H3
SCHEMBL17974909 0.75 NR1H2 (0.44) ALDH1A1TSHRPTPN1NR1H2NR1H3
SCHEMBL20945461 0.74 NR1H2 (0.58) NR1H2MAPT
SCHEMBL28135290 0.73 TSHR (0.46) ALDH1A1TSHRPTPN1ATMCYP2D6
SCHEMBL5709190 0.73 KCNN4 (0.46) ALDH1A1TSHRPTPN1ATMCYP2D6
SCHEMBL8755619 0.72 ALDH1A1 (0.41) ALDH1A1TSHRATMCYP2D6DRD2
SCHEMBL639889 0.72 ATM (0.41) ALDH1A1TSHRPTPN1ATMCYP2D6
SCHEMBL6846624 0.72 ATM (0.41) ALDH1A1TSHRPTPN1ATMCYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 15 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
JP-1225497-A None JP disclosed
US-8614081-B2 Nitrilase biocatalysts CODEXIS, INC. (US) 2013-12-24 US disclosed
US-20120142063-A1 NITRILASE BIOCATALYSTS Codexis ,Inc. (US) 2012-06-07 US disclosed
US-20120142063-A1 NITRILASE BIOCATALYSTS Codexis ,Inc. (US) 2012-06-07 US disclosed
US-20120142063-A1 NITRILASE BIOCATALYSTS Codexis ,Inc. (US) 2012-06-07 US disclosed
WO-2011011630-A2 NITRILASE BIOCATALYSTS CODEXIS, INC. (US) 2011-01-27 WO disclosed
WO-2011011630-A2 NITRILASE BIOCATALYSTS CODEXIS, INC. (US) 2011-01-27 WO disclosed
CN-101426769-A Five-membered heterocyclic invertebrate pest control agents DU PONT (US) 2009-05-06 CN disclosed
US-7414078-B2 Oral general anesthetics and metabolitically resistant anticonvulsants UNIVERSITY OF VIRGINIA PATENT FOUNDATION (US) 2008-08-19 US disclosed
US-7414078-B2 Oral general anesthetics and metabolitically resistant anticonvulsants UNIVERSITY OF VIRGINIA PATENT FOUNDATION (US) 2008-08-19 US disclosed
EP-0681713-B1 SULPHONIC ACID ESTERS, RADIATION-SENSITIVE MIXTURES MADE THEREWITH, AND THEIR USE CLARIANT GMBH (DE) 1998-11-18 EP disclosed
US-5716756-A POSITIVE OR NEGATIVE WORKING MIXTURES HOECHST AKTIENGESELLSCHAFT (DE) 1998-02-10 US disclosed
EP-0681713-A1 SULPHONIC ACID ESTERS, RADIATION-SENSITIVE MIXTURES MADE THEREWITH, AND THEIR USE HOECHST AKTIENGESELLSCHAFT (DE) 1995-11-15 EP disclosed
WO-1994018606-A1 SULPHONIC ACID ESTERS, RADIATION-SENSITIVE MIXTURES MADE THEREWITH, AND THEIR USE HOESCHT AKTIENGESELLSCHAFT (DE) 1994-08-18 WO disclosed
JP-H01225497-A PRODUCTION OF CARBOXYLIC ACID ESTER OF OPTICALLY ACTIVE FLUORINE-CONTAINING CYANOHYDRIN CENTRAL GLASS CO LTD 1989-09-08 JP disclosed