SCHEMBL9977537

SCHEMBL9977537

CCc1ccc(CN2CCN(Cc3ccc(C(C)(C)C)cc3)C2=O)cc1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 4/20 0.50
MEN1 O00255 2/20 0.50
ALDH1A1 P00352 1/20 0.50
POLB P06746 4/20 0.47
LMNA P02545 1/20 0.47
HDAC6 Q9UBN7 1/20 0.46
ERCC1 P07992 1/20 0.43
ERCC4 Q92889 1/20 0.43
CYP2D6 P10635 1/20 0.43
CYP2C9 P11712 1/20 0.43
CYP2C19 P33261 1/20 0.43
MGLL Q99685 1/20 0.42
RAB9A P51151 1/20 0.42
MAOB P27338 1/20 0.42
METAP2 P50579 1/20 0.40
DRD3 P35462 3/20 0.40
KCNH2 Q12809 3/20 0.40
HDAC1 Q13547 1/20 0.40
TDP1 Q9NUW8 1/20 0.40
DRD2 P14416 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9977538 0.93 POLB (0.51) KMT2AMEN1ALDH1A1POLBLMNA
SCHEMBL4606687 0.86 LMNA (0.46) KMT2AMEN1ALDH1A1POLBLMNA
SCHEMBL4595576 0.80 MAOB (0.47) KMT2AMEN1ALDH1A1POLBLMNA
SCHEMBL4595797 0.79 TRPV1 (0.54)
SCHEMBL4923161 0.79 HDAC6 (0.40) KMT2AMEN1ALDH1A1POLBLMNA
SCHEMBL10278887 0.78 MAOB (0.46) KMT2AMEN1ALDH1A1POLBLMNA
SCHEMBL4594671 0.78 KMT2A (0.47) KMT2AMEN1POLBLMNACYP2D6
SCHEMBL338386 0.76 BCHE (0.52) LMNAKCNH2
SCHEMBL3554203 0.76 RAB9A (0.58) KMT2AMEN1ALDH1A1HDAC6RAB9A
SCHEMBL4872875 0.76 MAPT (0.51) KMT2AMEN1ALDH1A1LMNAMGLL

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1874733-B1 SUBSTITUTED CYCLIC UREA DERIVATIVES AND THE USE THEREOF AS VANILLOID RECEPTOR 1 MODULATORS GRUENENTHAL GMBH (DE) 2012-06-20 EP disclosed