SCHEMBL9978290

SCHEMBL9978290

CNS(=O)(=O)c1ccc(OC(C)CC(F)(F)F)c([N+](=O)[O-])c1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
VCAM1 P19320 1/20 0.49
ALDH3A1 P30838 5/20 0.47
LMNA P02545 1/20 0.44
MAPT P10636 1/20 0.44
ALDH1A1 P00352 6/20 0.43
EPAS1 Q99814 1/20 0.41
PTPN1 P18031 1/20 0.40
HTT P42858 1/20 0.40
POLB P06746 1/20 0.40
TNNI3K Q59H18 2/20 0.40
BRAF P15056 1/20 0.40
CA12 O43570 1/20 0.40
CA1 P00915 1/20 0.40
CA2 P00918 1/20 0.40
CA3 P07451 1/20 0.40
CA4 P22748 1/20 0.40
CA6 P23280 1/20 0.40
CA5A P35218 1/20 0.40
CA7 P43166 1/20 0.40
CA9 Q16790 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12067076 0.85 VCAM1 (0.53) VCAM1ALDH3A1LMNAMAPTALDH1A1
SCHEMBL6912644 0.82 VCAM1 (0.58) VCAM1ALDH3A1LMNAMAPTALDH1A1
SCHEMBL12065563 0.82 POLB (0.44) LMNAPOLBTNNI3KBRAFCA1
SCHEMBL2278928 0.81 VCAM1 (0.53) VCAM1ALDH3A1LMNAMAPTALDH1A1
SCHEMBL12067917 0.80 VCAM1 (0.56) VCAM1ALDH3A1LMNAMAPTALDH1A1
SCHEMBL12067872 0.79 VCAM1 (0.57) VCAM1ALDH3A1LMNAMAPTALDH1A1
SCHEMBL15646981 0.78 IDH2 (0.52) VCAM1ALDH3A1ALDH1A1PTPN1HTT
SCHEMBL30871305 0.76 ALDH1A1 (0.67) VCAM1ALDH3A1LMNAMAPTALDH1A1
SCHEMBL6117960 0.76 ALDH1A1 (0.67) VCAM1ALDH3A1LMNAMAPTALDH1A1
SCHEMBL12065809 0.70 VCAM1 (0.47) VCAM1ALDH3A1LMNAMAPTALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011149827-A1 COMPOUNDS AND METHODS GLAXOSMITHKLINE LLC (US) 2011-12-01 WO disclosed
WO-2011149827-A1 COMPOUNDS AND METHODS GLAXOSMITHKLINE LLC (US) 2011-12-01 WO disclosed