SCHEMBL9978293

SCHEMBL9978293

CC#CCN(CC(=O)O)C(C)=O

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CHRM1 P11229 5/20 0.33
CHRM2 P08172 5/20 0.33
CHRM4 P08173 4/20 0.33
CHRM5 P08912 4/20 0.33
CHRM3 P20309 4/20 0.33
TDP1 Q9NUW8 2/20 0.31
EYA2 O00167 1/20 0.31
APP P05067 1/20 0.31
ACE P12821 1/20 0.31
KDM4E B2RXH2 1/20 0.30
LMNA P02545 1/20 0.30
ADRA2A P08913 1/20 0.30
ALOX15 P16050 1/20 0.30
TSHR P16473 1/20 0.30
DRD1 P21728 1/20 0.30
SLC6A2 P23975 1/20 0.30
SLC6A4 P31645 1/20 0.30
CYP2C19 P33261 1/20 0.30
ADRA1A P35348 1/20 0.30
DRD3 P35462 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9978268 0.79 MGAM (0.40) CHRM1CHRM2CHRM4CHRM5CHRM3
SCHEMBL468463 0.77 KDM4E (0.34) CHRM1CHRM2CHRM4CHRM5CHRM3
SCHEMBL2687920 0.77 TDP1 (0.43) CHRM2TDP1EYA2APPACE
SCHEMBL7421637 0.74 CTSK (0.35)
Water SCHEMBL7765711 0.74 TDP1 (0.41) CHRM2TDP1EYA2APPACE
SCHEMBL6788905 0.74 TDP1 (0.41) CHRM2TDP1EYA2APPACE
Water SCHEMBL7765705 0.74 TDP1 (0.41) CHRM2TDP1EYA2APPACE
SCHEMBL29956065 0.74 PYCR1 (0.36) CHRM1CHRM2CHRM4CHRM5CHRM3
SCHEMBL3714284 0.70 LMNA (0.39) CHRM1CHRM2CHRM4CHRM5CHRM3
SCHEMBL7975927 0.70 TDP1 (0.38) CHRM2TDP1EYA2APPACE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2576588-A1 METHODS FOR THE SYNTHESIS OF ALKYNE-CONTAINING DICARBA BRIDGES IN PEPTIDES Syngene Limited (AU) 2013-04-10 EP disclosed
WO-2011146974-A1 METHODS FOR THE SYNTHESIS OF ALKYNE-CONTAINING DICARBA BRIDGES IN PEPTIDES MONASH UNIVERSITY (AU) 2011-12-01 WO disclosed