SCHEMBL9979900

SCHEMBL9979900

CSCCCn1c(Cn2c(=O)[nH]c3ccncc32)nc2cc(Br)ccc21

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 4/20 0.36
TSHR P16473 2/20 0.36
MAPK1 P28482 2/20 0.36
HTT P42858 2/20 0.36
RECQL P46063 1/20 0.36
CYP3A4 P08684 2/20 0.35
ALDH1A1 P00352 2/20 0.34
SMN1; SMN2 Q16637 2/20 0.34
DAO P14920 1/20 0.34
LMNA P02545 1/20 0.34
HPGD P15428 1/20 0.34
TDP1 Q9NUW8 1/20 0.34
GABRA1 P14867 1/20 0.32
GABRA5 P31644 1/20 0.32
MEN1 O00255 1/20 0.32
CYP1A2 P05177 1/20 0.32
CYP2D6 P10635 1/20 0.32
CYP2C9 P11712 1/20 0.32
PKM P14618 1/20 0.32
CYP2C19 P33261 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15306210 0.79 CYP3A4 (0.60) MAPTCYP3A4ALDH1A1SMN1; SMN2CYP2D6
SCHEMBL16809273 0.76 CYP3A4 (0.38) CYP3A4
SCHEMBL9979897 0.73 LMNA (0.49) MAPK1ALDH1A1SMN1; SMN2LMNAMEN1
SCHEMBL17613273 0.69 CYP3A4 (0.60) CYP3A4CYP2D6
SCHEMBL30110668 0.66 CYP3A4 (0.59) CYP3A4
SCHEMBL9940698 0.66 CYP3A4 (0.59) CYP3A4
SCHEMBL16696095 0.66 TBXAS1 (0.36) HTTALDH1A1DAOLMNA
SCHEMBL6276891 0.66 CNR2 (0.40)
SCHEMBL9979857 0.65 CYP3A4 (0.62) RECQLCYP3A4CYP2D6
SCHEMBL6247536 0.65 CNR2 (0.37) TSHRMAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012080446-A1 BENZIMIDAZOLE RESPIRATORY SYNCYTIAL VIRUS INHIBITORS JANSSEN R&D IRELAND (IE) 2012-06-21 WO disclosed