SCHEMBL9980393

SCHEMBL9980393

NS(=O)(=O)c1ccc(CF)c(Nc2ncnc3[nH]nc(Br)c23)c1

nearest known ligand 0.40

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
TNNI3K Q59H18 14/20 0.40
BRAF P15056 6/20 0.40
CCNA2 P20248 2/20 0.34
CDK2 P24941 2/20 0.34
CDK1 P06493 1/20 0.34
CCNB1 P14635 1/20 0.34
CCNE1 P24864 1/20 0.34
CDK5 Q00535 1/20 0.34
CDK5R1 Q15078 1/20 0.34
CCNA1 P78396 1/20 0.33
CA1 P00915 1/20 0.33
CA2 P00918 1/20 0.33
ROCK1 Q13464 1/20 0.33
EGFR P00533 1/20 0.33
MKNK1 Q9BUB5 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9980396 0.87 TNNI3K (0.44) TNNI3KBRAFEGFR
SCHEMBL12067916 0.74 TNNI3K (0.62) TNNI3KBRAF
SCHEMBL12067874 0.72 TNNI3K (0.63) TNNI3KBRAF
SCHEMBL9980375 0.71 TNNI3K (0.40) TNNI3KBRAFCA1CA2
SCHEMBL9986097 0.71 TNNI3K (0.73) TNNI3KBRAF
SCHEMBL12067929 0.71 TNNI3K (0.57) TNNI3KBRAF
SCHEMBL12065804 0.71 TNNI3K (0.57) TNNI3KBRAF
SCHEMBL12065794 0.69 TNNI3K (0.50) TNNI3KBRAFMKNK1
SCHEMBL12065559 0.69 TNNI3K (0.50) TNNI3KBRAF
SCHEMBL9980436 0.68 TNNI3K (0.37) TNNI3KBRAFCA1CA2EGFR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011149827-A1 COMPOUNDS AND METHODS GLAXOSMITHKLINE LLC (US) 2011-12-01 WO disclosed