SCHEMBL9980599

SCHEMBL9980599

NC(=O)c1nc(N2CCCCC2)cn1-c1ccccc1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 2/20 0.44
HPGD P15428 6/20 0.44
ALDH1A1 P00352 5/20 0.44
HSD17B10 Q99714 5/20 0.44
TSHR P16473 3/20 0.44
KDM4E B2RXH2 3/20 0.44
GAA P10253 2/20 0.44
CASP1 P29466 1/20 0.44
CASP7 P55210 1/20 0.44
POLB P06746 1/20 0.42
ALOX12 P18054 1/20 0.42
PARP1 P09874 2/20 0.41
MAOB P27338 2/20 0.40
HTT P42858 3/20 0.40
SMN1; SMN2 Q16637 3/20 0.40
LMNA P02545 2/20 0.40
MEN1 O00255 2/20 0.40
KMT2A Q03164 2/20 0.40
USP2 O75604 1/20 0.40
MAPT P10636 3/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5365792 0.74 KDM4E (0.49) HPGDALDH1A1HSD17B10TSHRKDM4E
SCHEMBL5366159 0.73 HPGD (0.49) NPC1HPGDALDH1A1HSD17B10TSHR
Urea SCHEMBL27797099 0.72 NPC1 (0.61) NPC1HPGDALDH1A1HSD17B10TSHR
Carbamic Acid SCHEMBL27930251 0.72 NPC1 (0.61) NPC1HPGDALDH1A1HSD17B10TSHR
SCHEMBL5365804 0.72 KDM4E (0.47) HPGDALDH1A1HSD17B10TSHRKDM4E
SCHEMBL5374606 0.71 KMT2A (0.49) HPGDHSD17B10TSHRHTTSMN1; SMN2
SCHEMBL4553234 0.71 PTGS2 (0.48) GAAPOLBMAPK1
SCHEMBL9980597 0.69 ALDH1A1 (0.53) NPC1HPGDALDH1A1HSD17B10TSHR
SCHEMBL10002521 0.67 HSD11B1 (0.58) NPC1HPGDALDH1A1HSD17B10TSHR
Oxalic Acid SCHEMBL28160737 0.67 MAPT (0.63) NPC1HPGDALDH1A1HSD17B10TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2627650-A2 N-PHENYL IMIDAZOLE CARBOXAMIDE INHIBITORS OF 3-PHOSPHOINOSITIDE-DEPENDENT PROTEIN KINASE-1 Merck Sharp & Dohme Corp. (US) 2013-08-21 EP disclosed
WO-2011149874-A2 N-PHENYL IMIDAZOLE CARBOXAMIDE INHIBITORS OF 3-PHOSPHOINOSITIDE-DEPENDENT PROTEIN KINASE-1 SCHERING CORPORATION (US) 2011-12-01 WO disclosed