SCHEMBL998164

SCHEMBL998164

O=C(c1nccc(N2CCCC(O)C2)c1C1CC1)N(c1ccccc1)c1nnc[nH]1

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ROCK1 Q13464 3/20 0.37
CDC42BPB Q9Y5S2 3/20 0.37
ROCK2 O75116 2/20 0.37
PDE10A Q9Y233 4/20 0.34
SMARCA2 P51531 1/20 0.33
SMARCA4 P51532 1/20 0.33
PBRM1 Q86U86 1/20 0.33
PBK Q96KB5 1/20 0.33
LRRK2 Q5S007 1/20 0.32
MAPT P10636 2/20 0.31
LMNA P02545 1/20 0.31
MAPK1 P28482 1/20 0.31
HSD17B10 Q99714 1/20 0.31
KCNMA1 Q12791 1/20 0.31
IRAK4 Q9NWZ3 1/20 0.30
CCNE2 O96020 1/20 0.30
CCNE1 P24864 1/20 0.30
CDK2 P24941 1/20 0.30
GAA P10253 1/20 0.30
HPGD P15428 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL978875 0.74 HCAR2 (0.35) PDE10A
SCHEMBL992381 0.73 P2RX7 (0.31)
SCHEMBL980672 0.68 PTGIR (0.35) MAPTSMN1; SMN2
SCHEMBL986289 0.65 HDAC6 (0.43) MAPTLMNAHSD17B10GAAHPGD
SCHEMBL979099 0.64 NPSR1 (0.35) MAPTLMNAHSD17B10SMN1; SMN2
SCHEMBL1905179 0.64 PIM1 (0.49) MAPTMAPK1GAASMN1; SMN2
SCHEMBL15153028 0.63 HCAR2 (0.32)
SCHEMBL998166 0.62 PDE10A (0.36) PDE10ASMARCA2SMARCA4PBRM1LRRK2
SCHEMBL15405753 0.62 KCNMA1 (0.44) ROCK1CDC42BPBROCK2PDE10ASMARCA2
SCHEMBL977783 0.60 S1PR3 (0.33)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011008709-A1 APOPTOSIS SIGNAL-REGULATING KINASE INHIBITORS GILEAD SCIENCES, INC. (US) 2011-01-20 WO disclosed