SCHEMBL998194

SCHEMBL998194

COc1ccc(/C=C/C(=O)c2cc3c(cc2OCCN2CCOCC2)OCO3)cc1F

nearest known ligand 0.54

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
HIF1AN Q9NWT6 8/20 0.54
SMN1; SMN2 Q16637 3/20 0.51
KDM4E B2RXH2 4/20 0.50
MAPT P10636 4/20 0.50
ALDH1A1 P00352 3/20 0.50
RECQL P46063 1/20 0.50
ABCG2 Q9UNQ0 1/20 0.50
KEAP1 Q14145 2/20 0.49
NFE2L2 Q16236 2/20 0.49
LMNA P02545 1/20 0.48
TUBB1 Q9H4B7 1/20 0.47
MAPK1 P28482 1/20 0.47
HTT P42858 1/20 0.47
CYP3A4 P08684 2/20 0.47
CYP2D6 P10635 2/20 0.47
CYP2C9 P11712 2/20 0.47
CYP2C19 P33261 2/20 0.47
TSHR P16473 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL998195 1.00 HIF1AN (0.54) HIF1ANSMN1; SMN2KDM4EMAPTALDH1A1
SCHEMBL996376 0.93 HIF1AN (0.53) HIF1ANMAPTALDH1A1ABCG2TUBB1
SCHEMBL996379 0.93 HIF1AN (0.53) HIF1ANMAPTALDH1A1ABCG2TUBB1
SCHEMBL998223 0.92 HIF1AN (0.54) HIF1ANMAPTALDH1A1ABCG2TUBB1
SCHEMBL998221 0.92 HIF1AN (0.54) HIF1ANMAPTALDH1A1ABCG2TUBB1
SCHEMBL998259 0.89 KEAP1 (0.59) HIF1ANSMN1; SMN2KDM4EMAPTALDH1A1
SCHEMBL998257 0.89 KEAP1 (0.59) HIF1ANSMN1; SMN2KDM4EMAPTALDH1A1
SCHEMBL997051 0.88 TUBB1 (0.58) HIF1ANSMN1; SMN2KDM4EMAPTALDH1A1
SCHEMBL997056 0.88 TUBB1 (0.58) HIF1ANSMN1; SMN2KDM4EMAPTALDH1A1
SCHEMBL998657 0.87 HIF1AN (0.51) HIF1ANSMN1; SMN2KDM4EMAPTALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011009826-A2 NOVEL CHALCONE DERIVATIVES WITH CYTOTOXIC ACTIVITY ADAMED Sp.z o.o. (PL) 2011-01-27 WO disclosed