SCHEMBL998259

SCHEMBL998259

COc1ccc(C=CC(=O)c2cc3c(cc2OCCN2CCOCC2)OCO3)cc1

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KEAP1 Q14145 3/20 0.59
NFE2L2 Q16236 3/20 0.59
MAPT P10636 3/20 0.58
KDM4E B2RXH2 2/20 0.58
SMN1; SMN2 Q16637 2/20 0.58
MEN1 O00255 1/20 0.58
NPC1 O15118 1/20 0.58
GAA P10253 1/20 0.58
PKM P14618 1/20 0.58
RAB9A P51151 1/20 0.58
KMT2A Q03164 1/20 0.58
ALDH1A1 P00352 2/20 0.54
RECQL P46063 1/20 0.54
CYP3A4 P08684 1/20 0.52
CYP2D6 P10635 1/20 0.52
CYP2C9 P11712 1/20 0.52
TSHR P16473 1/20 0.52
CYP2C19 P33261 1/20 0.52
HIF1AN Q9NWT6 2/20 0.52
DRD2 P14416 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL998257 1.00 KEAP1 (0.59) KEAP1NFE2L2MAPTKDM4ESMN1; SMN2
SCHEMBL997108 0.93 MAPT (0.60) KEAP1NFE2L2MAPTKDM4ESMN1; SMN2
SCHEMBL997110 0.93 MAPT (0.60) KEAP1NFE2L2MAPTKDM4ESMN1; SMN2
SCHEMBL998730 0.92 MAPT (0.59) MAPTKDM4ESMN1; SMN2MEN1NPC1
SCHEMBL998727 0.92 MAPT (0.59) MAPTKDM4ESMN1; SMN2MEN1NPC1
SCHEMBL998194 0.89 HIF1AN (0.54) KEAP1NFE2L2MAPTKDM4ESMN1; SMN2
SCHEMBL998195 0.89 HIF1AN (0.54) KEAP1NFE2L2MAPTKDM4ESMN1; SMN2
SCHEMBL996808 0.88 KDM4E (0.56) KEAP1NFE2L2MAPTKDM4ESMN1; SMN2
SCHEMBL996811 0.88 KDM4E (0.56) KEAP1NFE2L2MAPTKDM4ESMN1; SMN2
SCHEMBL996636 0.87 TUBB4A (0.70) KEAP1NFE2L2MAPTKDM4ESMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011009826-A2 NOVEL CHALCONE DERIVATIVES WITH CYTOTOXIC ACTIVITY ADAMED Sp.z o.o. (PL) 2011-01-27 WO claimed
WO-2011009826-A2 NOVEL CHALCONE DERIVATIVES WITH CYTOTOXIC ACTIVITY ADAMED Sp.z o.o. (PL) 2011-01-27 WO disclosed