SCHEMBL9983137

SCHEMBL9983137

CCCc1ncc2cn[nH]c2n1

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.37
PDK2 Q15119 3/20 0.33
JAK2 O60674 2/20 0.33
ROCK2 O75116 2/20 0.33
PIM1 P11309 2/20 0.33
GSK3B P49841 2/20 0.33
ADORA3 P0DMS8 2/20 0.33
AURKA O14965 1/20 0.33
DAPK3 O43293 1/20 0.33
CHEK2 O96017 1/20 0.33
CDK2 P24941 1/20 0.33
MARK3 P27448 1/20 0.33
GSK3A P49840 1/20 0.33
LIMK1 P53667 1/20 0.33
CDK5 Q00535 1/20 0.33
ROCK1 Q13464 1/20 0.33
DYRK1A Q13627 1/20 0.33
AURKB Q96GD4 1/20 0.33
PRKD2 Q9BZL6 1/20 0.33
HTT P42858 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3260370 0.87 XDH (0.39) ALDH1A1ADORA3AGTR1AGTR2
SCHEMBL4566029 0.86 XDH (0.41) ALDH1A1HPGD
SCHEMBL4927108 0.84 ALDH1A1 (0.35) ALDH1A1ADORA3AURKACDK2HTT
SCHEMBL2555553 0.77 ALDH1A1 (0.33) ALDH1A1KDM4E
SCHEMBL7491917 0.72 ADORA3 (0.31) ALDH1A1JAK2ROCK2PIM1GSK3B
SCHEMBL11066168 0.70 PDK2 (0.35) ALDH1A1PDK2HPGDPDK4KDM4E
SCHEMBL479504 0.70 CYP1A2 (0.37) ALDH1A1JAK2ROCK2AURKADAPK3
SCHEMBL9983243 0.69 S1PR1 (0.32)
SCHEMBL9982977 0.69 HTR2C (0.47) JAK2ROCK2PIM1GSK3BAURKA
SCHEMBL3181459 0.69 PDK2 (0.38) ALDH1A1PDK2AURKACDK2HTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8076338-B2 Such as 6-(4-phenylpiperazin-1-yl)-9H-purine; cell proliferation/differentiation EXELIXIS, INC. (US) 2011-12-13 US disclosed