SCHEMBL9984601

SCHEMBL9984601

O=C(OCc1ccccc1)N1C(=O)OC2(CCNCC2)c2ccc(Cl)nc21

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
P2RX4 Q99571 3/20 0.37
P2RX1 P51575 1/20 0.37
P2RX3 P56373 1/20 0.37
HTR2C P28335 1/20 0.36
CTRB1 P17538 1/20 0.36
SLC29A1 Q99808 1/20 0.36
NPC1 O15118 1/20 0.36
GAA P10253 1/20 0.36
MAPK1 P28482 1/20 0.36
RAB9A P51151 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
TACR1 P25103 2/20 0.35
SLC6A4 P31645 1/20 0.35
KCNH2 Q12809 1/20 0.35
MEN1 O00255 1/20 0.35
KMT2A Q03164 1/20 0.35
NPSR1 Q6W5P4 1/20 0.35
GLA P06280 1/20 0.34
DDB1 Q16531 1/20 0.33
CRBN Q96SW2 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2525906 0.79 KCNH2 (0.48) HTR2CNPC1GAARAB9ASMN1; SMN2
SCHEMBL2526690 0.76 MEN1 (0.41) NPC1GAARAB9ASMN1; SMN2KCNH2
SCHEMBL1813226 0.72 KCNH2 (0.46) NPC1GAARAB9ASMN1; SMN2KCNH2
SCHEMBL31185337 0.72 KCNH2 (0.46) NPC1GAARAB9ASMN1; SMN2KCNH2
SCHEMBL28648250 0.67 CTRB1 (0.48) P2RX4P2RX1P2RX3HTR2CCTRB1
SCHEMBL18251771 0.65 GRM5 (0.42) HTR2CTACR1
SCHEMBL7711512 0.64 ENPP2 (0.54) HTR2CNPC1GAAMAPK1RAB9A
SCHEMBL30484110 0.63 MEN1 (0.57) NPC1MAPK1RAB9ASMN1; SMN2MEN1
SCHEMBL27193593 0.63 HTR2C (0.48) HTR2CNPC1GAAMAPK1RAB9A
SCHEMBL21800290 0.63 ABHD6 (0.55) HTR2CNPC1RAB9ASMN1; SMN2SLC6A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1861399-B1 CGRP RECEPTOR ANTAGONISTS MERCK SHARP & DOHME (US) 2011-12-14 EP disclosed