SCHEMBL9986996

SCHEMBL9986996

C=COc1cccc(C(=O)Oc2ccccc2)c1

nearest known ligand 0.51

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
MAPT P10636 6/20 0.51
TDP1 Q9NUW8 3/20 0.51
NSD2 O96028 1/20 0.50
MAPK1 P28482 1/20 0.50
ALDH1A1 P00352 4/20 0.48
ESR1 P03372 2/20 0.48
ESR2 Q92731 2/20 0.48
KMT2A Q03164 7/20 0.47
MEN1 O00255 2/20 0.47
PARP10 Q53GL7 1/20 0.46
ALOX5 P09917 1/20 0.45
RAB9A P51151 1/20 0.45
AKR1C3 P42330 1/20 0.45
SERPINE1 P05121 1/20 0.44
GALR1 P47211 1/20 0.44
L3MBTL1 Q9Y468 1/20 0.44
PKM P14618 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9986884 0.90 KMT2A (0.54) MAPTTDP1NSD2ALDH1A1ESR1
SCHEMBL5245757 0.83 L3MBTL1 (0.57) TDP1MAPK1ALDH1A1KMT2AMEN1
SCHEMBL69684 0.82 NSD2 (0.63) MAPTTDP1NSD2MAPK1ALDH1A1
SCHEMBL755296 0.82 SMN1; SMN2 (0.52) MAPTMAPK1ALDH1A1ESR1ESR2
SCHEMBL28168705 0.81 NSD2 (0.61) MAPTTDP1NSD2MAPK1ALDH1A1
SCHEMBL8673010 0.81 NSD2 (0.61) MAPTTDP1NSD2MAPK1ALDH1A1
SCHEMBL4357355 0.81 MAPT (0.51) MAPTTDP1NSD2MAPK1ALDH1A1
SCHEMBL10664572 0.79 PARP10 (0.65) MAPTTDP1NSD2MAPK1ALDH1A1
SCHEMBL11215809 0.78 AKR1C3 (0.68) MAPTTDP1NSD2MAPK1ALDH1A1
SCHEMBL28519972 0.78 ESR1 (0.73) MAPTTDP1NSD2ESR1ESR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011158149-A1 2-(3,5-DISUBSTITUTEDPHENYL)PYRIMIDIN-4(3H)-ONE DERIVATIVES PFIZER INC. (US) 2011-12-22 WO disclosed