SCHEMBL996213

SCHEMBL996213

CCOC[C@@H](Oc1ccc(C(F)(F)F)cc1)N1CCCC1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SLC6A4 P31645 7/20 0.42
LTA4H P09960 1/20 0.40
HTR6 P50406 3/20 0.39
HTR7 P34969 2/20 0.39
HTR1A P08908 2/20 0.39
HRH3 Q9Y5N1 4/20 0.38
KDM4E B2RXH2 3/20 0.37
ALDH1A1 P00352 2/20 0.37
MMP2 P08253 1/20 0.37
MMP9 P14780 1/20 0.37
TACR1 P25103 1/20 0.35
SLC6A2 P23975 3/20 0.35
SLC6A3 Q01959 3/20 0.35
NPC1 O15118 2/20 0.35
CYP2D6 P10635 2/20 0.35
CYP2C19 P33261 2/20 0.35
MTOR P42345 2/20 0.35
RAB9A P51151 2/20 0.35
KCNK2 O95069 2/20 0.35
KCNH2 Q12809 2/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL996214 1.00 SLC6A4 (0.42) SLC6A4LTA4HHTR6HTR7HTR1A
SCHEMBL999410 0.85 LTA4H (0.43) LTA4HHTR6HTR7HTR1AHRH3
SCHEMBL999411 0.85 LTA4H (0.43) LTA4HHTR6HTR7HTR1AHRH3
SCHEMBL1002192 0.85 HTR7 (0.44) SLC6A4LTA4HHTR6HTR7HTR1A
SCHEMBL1002190 0.85 HTR7 (0.44) SLC6A4LTA4HHTR6HTR7HTR1A
SCHEMBL1002275 0.82 HTR7 (0.42) LTA4HHTR6HTR7HTR1AHRH3
SCHEMBL1002277 0.82 HTR7 (0.42) LTA4HHTR6HTR7HTR1AHRH3
SCHEMBL994992 0.81 SLC6A4 (0.48) SLC6A4LTA4HHTR6HTR1AHRH3
SCHEMBL998852 0.80 SLC6A4 (0.41) SLC6A4LTA4HHTR6HTR1AHRH3
SCHEMBL998851 0.80 SLC6A4 (0.41) SLC6A4LTA4HHTR6HTR1AHRH3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2456436-A1 3-PHENOXYMETHYLPYRROLIDINE COMPOUNDS Theravance, Inc. (US) 2012-05-30 EP disclosed
WO-2011011231-A1 3-PHENOXYMETHYLPYRROLIDINE COMPOUNDS THERAVANCE, INC. (US) 2011-01-27 WO disclosed