SCHEMBL9988642

SCHEMBL9988642

Cc1cccnc1-c1cc(CNC(=O)O)cn1S(=O)(=O)c1cccnc1

nearest known ligand 0.41

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
TSHR P16473 1/20 0.41
ALDH1A1 P00352 2/20 0.41
NAMPT P43490 10/20 0.39
IDE P14735 1/20 0.38
NOTUM Q6P988 1/20 0.38
KMT2A Q03164 1/20 0.38
LMNA P02545 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1581058 0.89 TSHR (0.38) TSHRALDH1A1KMT2A
Fumaric Acid SCHEMBL1278717 0.88 HDAC1 (0.35) TSHRALDH1A1NAMPTKMT2A
Fumaric Acid SCHEMBL1278719 0.88 HDAC1 (0.35) TSHRALDH1A1NAMPTKMT2A
SCHEMBL9989094 0.87 TSHR (0.42) TSHRALDH1A1NAMPTLMNA
SCHEMBL9989128 0.87 ALDH1A1 (0.43) TSHRALDH1A1NAMPTIDE
SCHEMBL3906007 0.86 TSHR (0.42) TSHRALDH1A1NAMPTLMNA
SCHEMBL9988058 0.83 CYP2C9 (0.40) TSHRALDH1A1NAMPTLMNA
SCHEMBL9988101 0.82 NAMPT (0.45) TSHRALDH1A1NAMPT
SCHEMBL4792179 0.81 CYP2A6 (0.36) TSHRALDH1A1IDE
SCHEMBL9989088 0.80 NTRK1 (0.46) TSHRALDH1A1NAMPTLMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8299261-B2 1-heterocyclylsulfonyl, 3-aminomethyl, 5-(hetero-) aryl substituted 1-H-pyrrole derivatives as acid secretion inhibitors TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2012-10-30 US disclosed
US-20110301173-A1 1-HETEROCYCLYLSULFONYL, 3-AMINOMETHYL, 5- (HETERO-) ARYL SUBSTITUTED 1-H-PYRROLE DERIVATIVES AS ACID SECRETION INHIBITORS TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2011-12-08 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20110301173-A1 1-HETEROCYCLYLSULFONYL, 3-AMINOMETHYL, 5- (HETERO-) ARYL SUBSTITUTED 1-H-PYRROLE DERIVATIVES AS ACID SECRETION INHIBITORS GHSR, HRH2, ASNS TSHR 287/4885ALDH1A1 1975/4885NAMPT 1948/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.