SCHEMBL9989128

SCHEMBL9989128

Cc1ccccc1-c1cc(CNC(=O)O)cn1S(=O)(=O)c1cccnc1

nearest known ligand 0.43

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.43
NAMPT P43490 10/20 0.42
TSHR P16473 1/20 0.42
CYP2C9 P11712 1/20 0.40
TP53 P04637 1/20 0.40
TDP1 Q9NUW8 1/20 0.39
IDE P14735 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3906007 0.93 TSHR (0.42) ALDH1A1NAMPTTSHRCYP2C9
SCHEMBL9989094 0.90 TSHR (0.42) ALDH1A1NAMPTTSHRCYP2C9TP53
SCHEMBL29754033 0.89 ALDH1A1 (0.39) ALDH1A1TSHR
SCHEMBL194035 0.89 ALDH1A1 (0.39) ALDH1A1TSHR
Hydrochloric Acid SCHEMBL1156606 0.88 ALDH1A1 (0.38) ALDH1A1TSHR
Fumaric Acid SCHEMBL194496 0.88 ALDH1A1 (0.37) ALDH1A1NAMPTTSHR
Fumaric Acid SCHEMBL194497 0.88 ALDH1A1 (0.37) ALDH1A1NAMPTTSHR
Fumaric Acid SCHEMBL29536757 0.88 ALDH1A1 (0.37) ALDH1A1NAMPTTSHR
SCHEMBL9988058 0.87 CYP2C9 (0.40) ALDH1A1NAMPTTSHRCYP2C9
SCHEMBL9988642 0.87 TSHR (0.41) ALDH1A1NAMPTTSHRIDE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8299261-B2 1-heterocyclylsulfonyl, 3-aminomethyl, 5-(hetero-) aryl substituted 1-H-pyrrole derivatives as acid secretion inhibitors TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2012-10-30 US disclosed
US-20110301173-A1 1-HETEROCYCLYLSULFONYL, 3-AMINOMETHYL, 5- (HETERO-) ARYL SUBSTITUTED 1-H-PYRROLE DERIVATIVES AS ACID SECRETION INHIBITORS TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2011-12-08 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20110301173-A1 1-HETEROCYCLYLSULFONYL, 3-AMINOMETHYL, 5- (HETERO-) ARYL SUBSTITUTED 1-H-PYRROLE DERIVATIVES AS ACID SECRETION INHIBITORS GHSR, HRH2, ASNS ALDH1A1 1975/4885NAMPT 1948/4885TSHR 287/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.