SCHEMBL9995371

SCHEMBL9995371

NC(=O)C(=COc1ccncn1)c1ccccc1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 3/20 0.40
RAB9A P51151 3/20 0.40
KMT2A Q03164 7/20 0.37
MEN1 O00255 1/20 0.37
PKM P14618 2/20 0.36
HTT P42858 1/20 0.36
GFER P55789 1/20 0.36
MITF O75030 1/20 0.36
CDK5 Q00535 1/20 0.36
CDK5R1 Q15078 1/20 0.36
TBXA2R P21731 4/20 0.35
ALDH1A1 P00352 4/20 0.34
CYP3A4 P08684 3/20 0.34
CYP2C19 P33261 3/20 0.34
CYP1A2 P05177 2/20 0.34
CYP2D6 P10635 2/20 0.34
CYP2C9 P11712 2/20 0.34
PLOD2 O00469 1/20 0.34
PLOD3 O60568 1/20 0.34
HPGD P15428 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21682467 0.78 NPC1 (0.40) NPC1RAB9AKMT2AMEN1PKM
SCHEMBL23422080 0.73 F7 (0.46) NPC1RAB9AKMT2AHTTALDH1A1
SCHEMBL15477869 0.72 KMT2A (0.48) NPC1RAB9AKMT2AMEN1PKM
Pyrimidine SCHEMBL25385683 0.71 KMT2A (0.44) NPC1RAB9AKMT2AMEN1ALDH1A1
SCHEMBL9995369 0.69 MCL1 (0.38) NPC1RAB9AKMT2APKMALDH1A1
SCHEMBL9995368 0.69 MCL1 (0.38) NPC1RAB9AKMT2APKMALDH1A1
SCHEMBL15175637 0.67 ALDH1A1 (0.39) KMT2AHTTALDH1A1CYP2C19HPGD
SCHEMBL8390998 0.67 HSP90AA1 (0.45) NPC1RAB9AKMT2AMEN1CYP3A4
SCHEMBL20995693 0.66 AKR1C1 (0.43) NPC1RAB9AKMT2AMEN1PKM
SCHEMBL3670626 0.66 CYP2C19 (0.50) KMT2AMEN1PKMHTTALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2585470-A2 NOVEL FUSED PYRIMIDINE DERIVATIVES FOR INHD3ITION OF TYROSINE KINASE ACTIVITY Hanmi Science Co., Ltd. (KR) 2013-05-01 EP disclosed
WO-2011162515-A2 NOVEL FUSED PYRIMIDINE DERIVATIVES FOR INHD3ITION OF TYROSINE KINASE ACTIVITY HANMI HOLDINGS CO. , LTD. (KR) 2011-12-29 WO disclosed