SCHEMBL10024019

SCHEMBL10024019

COC(=O)C(CO)NC(=O)c1ccccc1

nearest known ligand 0.56

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
GAA P10253 2/20 0.56
RAB9A P51151 1/20 0.56
ALDH1A1 P00352 3/20 0.55
LMNA P02545 1/20 0.55
GLA P06280 1/20 0.55
THRB P10828 1/20 0.51
CYP2C9 P11712 1/20 0.51
CYP2C19 P33261 1/20 0.51
HSD17B10 Q99714 1/20 0.51
CYP26A1 O43174 1/20 0.51
GPR139 Q6DWJ6 1/20 0.51
KMT2A Q03164 1/20 0.50
CTSL P07711 1/20 0.50
TAS1R3 Q7RTX0 4/20 0.49
TAS1R1 Q7RTX1 4/20 0.49
L3MBTL1 Q9Y468 1/20 0.48
CA2 P00918 2/20 0.48
CA1 P00915 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5672076 1.00 GAA (0.56) GAARAB9AALDH1A1LMNAGLA
SCHEMBL9925857 0.94 ALDH1A1 (0.56) GAARAB9AALDH1A1LMNAGLA
SCHEMBL26199837 0.87 CYP26A1 (0.53) GAARAB9AALDH1A1CYP26A1GPR139
SCHEMBL27673425 0.87 CYP26A1 (0.53) GAARAB9AALDH1A1CYP26A1GPR139
SCHEMBL3679721 0.87 RAB9A (0.59) GAARAB9AALDH1A1LMNAGLA
SCHEMBL23967346 0.85 GAA (0.54) GAARAB9AALDH1A1LMNAGLA
SCHEMBL7448811 0.85 GAA (0.54) GAARAB9AALDH1A1LMNAGLA
SCHEMBL7448810 0.85 GAA (0.54) GAARAB9AALDH1A1LMNAGLA
SCHEMBL8235468 0.85 CA1 (0.56) GAARAB9AALDH1A1LMNAGLA
SCHEMBL13885653 0.85 LNPEP (0.56) GAARAB9ATAS1R3TAS1R1L3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023130008-A2 PHARMACEUTICAL COMPOSITIONS OF 6-(2-(2H-TETRAZOL-5-YL)ETHYL)DECAHYDROISOQUINOLINE-3-CARBOXYLIC ACID AND DERIVATIVES THEREOF SEA PHARMACEUTICALS LLC (US) 2023-07-06 WO disclosed
EP-2957555-A1 METHOD FOR MODIFYING DERIVATIVES OF AMINO ACIDS AND PEPTIDES, COMPOUNDS PRODUCED, AND USE Consejo Superior De Investigaciones Científicas (CSIC) (ES) 2015-12-23 EP disclosed
WO-2014125145-A1 METHOD FOR MODIFYING DERIVATIVES OF AMINO ACIDS AND PEPTIDES, COMPOUNDS PRODUCED, AND USE CONSEJO SUPERIOR DE INVESTIGACIONES CIENTÍFICAS (CSIC) (ES) 2014-08-21 WO disclosed
WO-2013001120-A1 CHEMICAL PROCESS FOR THE SELECTIVE MODIFICATION OF PEPTIDES CONSEJO SUPERIOR DE INVESTIGACIONES CIENTÍFICAS (CSIC) (ES) 2013-01-03 WO disclosed
WO-2012017114-A1 METHOD FOR OBTAINING AZETIDINE DERIVATIVES CONSEJO SUPERIOR DE INVESTIGACIONES CIENTÍFICAS (CSIC) (ES) 2012-02-09 WO disclosed