SCHEMBL10033089

SCHEMBL10033089

C=C(C[C@@H]1CC[C@@H](N)[C@H](c2ccc(F)cc2F)C1)OCC

nearest known ligand 0.40

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 3/20 0.40
HTR2C P28335 2/20 0.40
HTR2B P41595 2/20 0.40
KDM1A O60341 8/20 0.38
KDM1B Q8NB78 3/20 0.38
GAA P10253 1/20 0.36
ALDH1A1 P00352 1/20 0.34
TDP1 Q9NUW8 1/20 0.34
OPRL1 P41146 1/20 0.34
NR3C2 P08235 1/20 0.34
DPP4 P27487 3/20 0.33
GPR88 Q9GZN0 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10033085 0.84 HTR2A (0.40) HTR2AHTR2CHTR2BKDM1AALDH1A1
SCHEMBL10033086 0.83 KDM1A (0.40) HTR2CHTR2BKDM1AKDM1BALDH1A1
SCHEMBL10033111 0.80 HTR2C (0.35) HTR2AHTR2CHTR2BGAAALDH1A1
SCHEMBL17806039 0.70 HTR2A (0.53) HTR2AHTR2CHTR2BKDM1AKDM1B
SCHEMBL15597453 0.70 KDM1A (0.71) HTR2AHTR2CHTR2BKDM1AKDM1B
SCHEMBL15541134 0.70 ALDH1A1 (0.48) HTR2AHTR2CHTR2BGAAALDH1A1
Hydrochloric Acid SCHEMBL16371833 0.69 HTR2A (0.56) HTR2AHTR2CHTR2BKDM1AKDM1B
SCHEMBL10032839 0.67 KDM1A (0.40) KDM1AKDM1BDPP4
SCHEMBL10032974 0.66 SIGMAR1 (0.44) HTR2CKDM1A
SCHEMBL10033088 0.66 KDM1A (0.34) KDM1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012046771-A1 CYCLOALKANE COMPOUND アステラス製薬株式会社 (JP) 2012-04-12 WO disclosed