SCHEMBL10033099

SCHEMBL10033099

COC(=O)CC1CCCC(N)C1c1ccc(C#N)cc1

nearest known ligand 0.40

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
CTSC P53634 5/20 0.40
HDAC8 Q9BY41 2/20 0.39
HDAC6 Q9UBN7 2/20 0.39
HDAC1 Q13547 1/20 0.39
KDM1A O60341 3/20 0.38
PAX8 Q06710 2/20 0.38
GRIA4 P48058 1/20 0.38
KCNH2 Q12809 3/20 0.38
HTT P42858 1/20 0.36
USP30 Q70CQ3 1/20 0.35
NPC1 O15118 1/20 0.35
RAB9A P51151 1/20 0.35
FASN P49327 1/20 0.35
EGLN1 Q9GZT9 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10033097 0.84 KDM4E (0.39) HDAC8HDAC6HDAC1
SCHEMBL10033109 0.84 KDM1A (0.41) HDAC8HDAC6HDAC1KDM1A
SCHEMBL10033125 0.79 GRIA4 (0.38) HDAC8HDAC6HDAC1KDM1AGRIA4
SCHEMBL1709398 0.79 KDM1A (0.36) HDAC8HDAC6HDAC1KDM1APAX8
SCHEMBL25222944 0.76 KDM1A (0.42) KDM1AGRIA4HTT
SCHEMBL10033104 0.72 MEN1 (0.38) HTTNPC1RAB9A
SCHEMBL10033130 0.70 TACR1 (0.41) KDM1A
SCHEMBL9166296 0.69 POLB (0.40)
SCHEMBL10033102 0.69 PTGDR (0.40)
Hydrochloric Acid SCHEMBL28795083 0.68 EPHX2 (0.38)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012046771-A1 CYCLOALKANE COMPOUND アステラス製薬株式会社 (JP) 2012-04-12 WO disclosed