SCHEMBL10033102

SCHEMBL10033102

COC(=O)CC1CCCC(N)C1c1ccc(Cl)cc1F

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGDR Q13258 1/20 0.40
PTGDR2 Q9Y5Y4 1/20 0.40
OPRL1 P41146 4/20 0.40
HTR2A P28223 1/20 0.38
HTR2C P28335 1/20 0.38
HTR2B P41595 1/20 0.38
ALDH1A1 P00352 1/20 0.36
L3MBTL1 Q9Y468 1/20 0.36
KMT2A Q03164 2/20 0.36
DPP4 P27487 2/20 0.34
MDM2 Q00987 2/20 0.34
TP53 P04637 1/20 0.34
ABL1 P00519 1/20 0.33
GPBAR1 Q8TDU6 1/20 0.33
PROKR1 Q8TCW9 1/20 0.33
CYP11B1 P15538 1/20 0.33
CYP11B2 P19099 1/20 0.33
MEN1 O00255 1/20 0.33
POLB P06746 1/20 0.33
TLR4 O00206 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10033097 0.81 KDM4E (0.39) PTGDRPTGDR2ALDH1A1MDM2POLB
SCHEMBL10033125 0.81 GRIA4 (0.38) HTR2AHTR2CHTR2B
SCHEMBL1709399 0.80 PTGDR (0.41) PTGDRPTGDR2OPRL1ALDH1A1L3MBTL1
SCHEMBL10033128 0.78 ALOX5AP (0.36) ALDH1A1L3MBTL1KMT2ADPP4CYP11B1
SCHEMBL10033098 0.74 ALOX5AP (0.39) ALDH1A1L3MBTL1DPP4CYP11B1CYP11B2
SCHEMBL10033129 0.74 PPOX (0.36) ALDH1A1L3MBTL1KMT2ADPP4CYP11B1
SCHEMBL10033100 0.74 CYP11B1 (0.35) ALDH1A1L3MBTL1DPP4CYP11B1CYP11B2
SCHEMBL10033112 0.73 BRD4 (0.42) ALDH1A1KMT2APOLB
SCHEMBL10033095 0.72 L3MBTL1 (0.41) ALDH1A1L3MBTL1KMT2ADPP4MEN1
SCHEMBL10033109 0.72 KDM1A (0.41) ALDH1A1KMT2APOLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012046771-A1 CYCLOALKANE COMPOUND アステラス製薬株式会社 (JP) 2012-04-12 WO disclosed