SCHEMBL1709398

SCHEMBL1709398

COC(=O)CC1CCCC(N(CC2CCCCC2)CC2CCCCC2)C1c1ccc(C#N)cc1

nearest known ligand 0.36

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
KDM1A O60341 5/20 0.36
TSHR P16473 2/20 0.35
USP30 Q70CQ3 1/20 0.35
NPC1 O15118 1/20 0.35
RAB9A P51151 1/20 0.35
EPHX1 P07099 1/20 0.34
KMT2A Q03164 1/20 0.34
GRIA4 P48058 1/20 0.33
PAX8 Q06710 1/20 0.33
ITK Q08881 1/20 0.33
NAMPT P43490 1/20 0.33
CTSD P07339 1/20 0.33
BACE1 P56817 1/20 0.33
HDAC8 Q9BY41 2/20 0.32
HDAC6 Q9UBN7 2/20 0.32
HDAC1 Q13547 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10033121 0.89 USP30 (0.38) KDM1ATSHRUSP30NPC1RAB9A
SCHEMBL10033001 0.87 NPC1 (0.38) NPC1RAB9AKMT2A
SCHEMBL10033003 0.87 EPHX2 (0.45) NPC1RAB9AKMT2A
SCHEMBL10033134 0.82 USP30 (0.36) KDM1AUSP30NPC1RAB9AGRIA4
SCHEMBL1709497 0.79 EPHX2 (0.43) USP30KMT2A
SCHEMBL10033099 0.79 CTSC (0.40) KDM1AUSP30NPC1RAB9AGRIA4
SCHEMBL10033135 0.78 KCNN4 (0.38) EPHX1CTSDHDAC8HDAC6HDAC1
SCHEMBL1709374 0.77 KMT2A (0.39) RAB9AKMT2A
SCHEMBL1709408 0.76 DGAT1 (0.38)
SCHEMBL1709407 0.76 TP53 (0.39) NPC1RAB9AEPHX1KMT2APAX8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012046771-A1 CYCLOALKANE COMPOUND アステラス製薬株式会社 (JP) 2012-04-12 WO disclosed