SCHEMBL10037140

SCHEMBL10037140

CC(C)N1CCN(Cc2cccc3ccccc23)CC1

nearest known ligand 0.62

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ACHE P22303 2/20 0.61
MC4R P32245 2/20 0.56
DRD2 P14416 2/20 0.53
DRD4 P21917 2/20 0.53
DRD3 P35462 2/20 0.53
FAAH O00519 1/20 0.51
MAPT P10636 4/20 0.50
PKM P14618 2/20 0.50
MAPK1 P28482 2/20 0.50
TDP1 Q9NUW8 2/20 0.50
MEN1 O00255 1/20 0.50
KMT2A Q03164 1/20 0.50
KDM4E B2RXH2 1/20 0.50
GAA P10253 1/20 0.50
ALDH1A1 P00352 1/20 0.49
GPR84 Q9NQS5 1/20 0.49
OPRL1 P41146 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3864845 0.82 FAAH (0.54) FAAHMEN1KMT2AKDM4EALDH1A1
SCHEMBL12123080 0.82 ACHE (0.67) ACHEMC4RDRD2DRD4DRD3
SCHEMBL11887347 0.82 ACHE (0.66) ACHEDRD2DRD4DRD3FAAH
SCHEMBL3921135 0.80 ACHE (0.68) ACHEDRD2DRD4DRD3FAAH
SCHEMBL31392633 0.80 ACHE (0.68) ACHEDRD2DRD4DRD3FAAH
SCHEMBL10701626 0.79 ACHE (0.62) ACHEDRD2DRD4DRD3FAAH
SCHEMBL15800713 0.79 ACHE (0.62) ACHEDRD2DRD4DRD3FAAH
SCHEMBL17460736 0.79 KMT2A (0.67) ACHEMAPTTDP1MEN1KMT2A
SCHEMBL807336 0.78 ACHE (0.66) ACHEDRD2DRD4DRD3FAAH
SCHEMBL31010166 0.78 ACHE (0.66) ACHEDRD2DRD4DRD3FAAH

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20120022070-A1 Heat Shock Protein 90 Inhibitors, Methods Of Preparing Same, And Methods For Their Use EMORY UNIVERSITY (US) 2012-01-26 US disclosed
US-20120022070-A1 Heat Shock Protein 90 Inhibitors, Methods Of Preparing Same, And Methods For Their Use EMORY UNIVERSITY (US) 2012-01-26 US disclosed
US-20110281908-A1 Aminoquinoline Derived Heat Shock Protein 90 Inhibitors, Methods Of Preparing Same, And Methods For Their Use EMORY UNIVERSITY (US) 2011-11-17 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20110281908-A1 Aminoquinoline Derived Heat Shock Protein 90 Inhibitors, Methods Of Preparing Same, And Methods For Their Use HSP90AB1, HSP90AB2P, HSP90AA1 ACHE 3037/4885MC4R 4580/4885DRD2 4546/4885
US-20120022070-A1 Heat Shock Protein 90 Inhibitors, Methods Of Preparing Same, And Methods For Their Use HSP90AB1, HSP90AA1, HSP90AB2P ACHE 3511/4885MC4R 4696/4885DRD2 4865/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.