SCHEMBL10044524

SCHEMBL10044524

COc1cc(C)c(OCC[S+](C)[O-])c(OC)c1

nearest known ligand 0.38

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
BRD4 O60885 3/20 0.38
CYP1A2 P05177 2/20 0.36
MAPK1 P28482 1/20 0.36
CRHR1 P34998 1/20 0.34
L3MBTL1 Q9Y468 4/20 0.33
MAPT P10636 3/20 0.33
PTPN1 P18031 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
CYP1A1 P04798 1/20 0.33
CYP1B1 Q16678 1/20 0.33
LMNA P02545 1/20 0.32
CYP19A1 P11511 1/20 0.32
NQO2 P16083 1/20 0.32
IL17A Q16552 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18639409 0.84 MAPK1 (0.47) BRD4CYP1A2MAPK1L3MBTL1MAPT
SCHEMBL15180031 0.81 CA1 (0.39) BRD4CYP1A2MAPK1CYP1A1CYP1B1
SCHEMBL10044605 0.78 BRD4 (0.55) BRD4CYP1A2MAPK1L3MBTL1MAPT
SCHEMBL10044945 0.75 L3MBTL1 (0.45) BRD4CYP1A2MAPK1L3MBTL1MAPT
SCHEMBL10044942 0.73 BRD4 (0.48) BRD4CYP1A2MAPK1L3MBTL1MAPT
SCHEMBL10044441 0.73 BRD4 (0.40) BRD4CYP1A2MAPK1L3MBTL1CYP1A1
SCHEMBL10044445 0.72 LMNA (0.48) BRD4CYP1A2PTPN1LMNA
SCHEMBL18292053 0.72 MAPK1 (0.58) BRD4CYP1A2MAPK1SMN1; SMN2CYP1A1
SCHEMBL684136 0.72 ACHE (0.52) CYP1A2MAPTPTPN1CYP1A1CYP1B1
SCHEMBL18292070 0.70 SMN1; SMN2 (0.59) BRD4CYP1A2MAPK1L3MBTL1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012052420-A1 METHOD FOR PREPARING SUBSTITUTED N-(3-AMINO-QUINOXALIN-2-YL)-SULFONAMIDES AND THEIR INTERMEDIATES N-(3-CHLORO-QUINOXALIN-2-YL)SULFONAMIDES MERCK SERONO S.A. GENEVA (CH) 2012-04-26 WO disclosed