SCHEMBL1004733

SCHEMBL1004733

CCCCCCCCCC(=O)OC(CO)COC(=O)CCCCCCC

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
PRKCA P17252 5/20 1.00
PRKCE Q02156 2/20 1.00
PRKCQ Q04759 2/20 1.00
PRKCD Q05655 2/20 1.00
ALDH1A1 P00352 1/20 0.84
LMNA P02545 1/20 0.84
MAPT P10636 1/20 0.77
MAPK1 P28482 1/20 0.77
LPAR3 Q9UBY5 3/20 0.67
LPAR1 Q92633 2/20 0.67
ENPP2 Q13822 1/20 0.67
SMN1; SMN2 Q16637 1/20 0.67
KDM4E B2RXH2 1/20 0.66
DUSP3 P51452 1/20 0.66
MEN1 O00255 1/20 0.66
KMT2A Q03164 1/20 0.66

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4176661 1.00 PRKCA (1.00) PRKCAPRKCEPRKCQPRKCDALDH1A1
SCHEMBL8049183 1.00 PRKCA (1.00) PRKCAPRKCEPRKCQPRKCDALDH1A1
SCHEMBL16431424 1.00 PRKCA (1.00) PRKCAPRKCEPRKCQPRKCDALDH1A1
SCHEMBL23992003 1.00 PRKCA (1.00) PRKCAPRKCEPRKCQPRKCDALDH1A1
SCHEMBL12171707 1.00 PRKCA (1.00) PRKCAPRKCEPRKCQPRKCDALDH1A1
SCHEMBL23668326 1.00 PRKCA (1.00) PRKCAPRKCEPRKCQPRKCDALDH1A1
SCHEMBL8388177 1.00 PRKCA (1.00) PRKCAPRKCEPRKCQPRKCDALDH1A1
SCHEMBL8048373 1.00 PRKCA (1.00) PRKCAPRKCEPRKCQPRKCDALDH1A1
SCHEMBL2502820 1.00 PRKCA (1.00) PRKCAPRKCEPRKCQPRKCDALDH1A1
SCHEMBL8384466 1.00 PRKCA (1.00) PRKCAPRKCEPRKCQPRKCDALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 90 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4724049-A1 MODIFIED RELEASE FILL COMPOSITIONS FOR DOSAGE FORMS AND METHODS OF PREPARATION AND USE THEREOF Catalent Ontario Limited (CA) 2026-04-15 EP claimed
US-20260042933-A1 Formulation For Simultaneous Rejuvenation And Protection Of The Interior Fibers And Exterior Surfaces Of Wood WINGET RICHARD (US) 2026-02-12 US claimed
CN-117717157-B Preparation method of transparent emulsified nano essence with low surfactant 嘉兴未来食品研究院 2025-05-09 CN claimed
WO-2024254056-A1 MODIFIED RELEASE FILL COMPOSITIONS FOR DOSAGE FORMS AND METHODS OF PREPARATION AND USE THEREOF CATALENT ONTARIO LIMITED (CA) 2024-12-12 WO claimed
US-11793754-B1 Sodium hypochlorite and chlorhexidine based nanoemulsions and a method of preparation thereof KING ABDULAZIZ UNIVERSITY (SA) 2023-10-24 US claimed
CN-116370345-A Transparent oil solution containing ceramide and sphingosine and preparation method thereof 重庆智合生物医药有限公司 2023-07-04 CN claimed
CN-116139082-A Self-microemulsion composition and preparation and application thereof 湖南慧泽生物医药科技有限公司 2023-05-23 CN claimed
EP-2525827-B1 PHARMACEUTICAL FORMULATIONS OF LORATADINE FOR ENCAPSULATION AND COMBINATIONS THEREOF CATALENT ONTARIO LTD (CA) 2020-11-18 EP claimed
EP-3653204-A1 PHARMACEUTICAL FORMULATIONS OF LORATADINE FOR ENCAPSULATION AND COMBINATIONS THEREOF Catalent Ontario Limited (CA) 2020-05-20 EP claimed
WO-2013008083-A1 PHARMACEUTICAL COMPOSITION FOR ENHANCING ANTICANCER EFFICACY OF TAMOXIFEN NATIONAL INSTITUTE OF PHARMACEUTICAL EDUCATION AND RESEARCH (NIPER) (IN) 2013-01-17 WO claimed
US-20120301544-A1 PHARMACEUTICAL FORMULATIONS OF LORATADINE FOR ENCAPSULATION AND COMBINATIONS THEREOF ACCUCAPS INDUSTRIES LIMITED (CA) 2012-11-29 US claimed
WO-2011088550-A1 PHARMACEUTICAL FORMULATIONS OF LORATADINE FOR ENCAPSULATION AND COMBINATIONS THEREOF ACCUCAPS INDUSTRIES LIMITED (CA) 2011-07-28 WO claimed
WO-2011004395-A1 MICROEMULSION FORMULATION FOR BIOLOGICALS INTAS BIOPHARMACEUTICALS LIMITED (IN) 2011-01-13 WO claimed
EP-0995430-A2 Use of diacylolycerols for enhancing the barrier function of the skin Beiersdorf Aktiengesellschaft (DE) 2000-04-26 EP claimed
EP-0655907-B1 USE OF DIACYLOLYCEROLS FOR INCREASING THE MELANIN CONTENT IN MELANOCYTES UNIV BOSTON (US) 1999-04-28 EP claimed
EP-0542108-B1 Stabilizers for plastic materials CIBA GEIGY AG (CH) 1997-09-24 EP claimed
EP-0730001-A1 Stabilizers for plastic materials F. HOFFMANN-LA ROCHE AG (CH) 1996-09-04 EP claimed
WO-1996009810-A1 METHODS FOR ENHANCING MELANIN SYNTHESIS IN MELANOCYTES USING DIACYLGLYCEROLS AND USES THEREOF TRUSTEES OF BOSTON UNIVERSITY (US) 1996-04-04 WO claimed
EP-0542108-A2 Stabilizers for plastic materials F. HOFFMANN-LA ROCHE AG (CH) 1993-05-19 EP claimed
JP-8245830-A None JP disclosed
EP-4724049-A1 MODIFIED RELEASE FILL COMPOSITIONS FOR DOSAGE FORMS AND METHODS OF PREPARATION AND USE THEREOF Catalent Ontario Limited (CA) 2026-04-15 EP disclosed
US-20260042933-A1 Formulation For Simultaneous Rejuvenation And Protection Of The Interior Fibers And Exterior Surfaces Of Wood WINGET RICHARD (US) 2026-02-12 US disclosed
US-20250213497-A1 A NANO IN MICRO FORMULATION AND PROCESS THEREOF AMRITA VISHWA VIDYAPEETHAM (IN) 2025-07-03 US disclosed
EP-3728487-B1 METHOD OF REMOVING POLYMERIC MATERIAL COMPRISING HETEROATOMS FROM A SURFACE USING COMPOSITIONS INCLUDING A KETO-ESTER COMPOUND FOURTH PRINCIPLE LLC (US) 2025-07-02 EP disclosed
CN-119264010-A Meta-diacyl compound and application thereof 河南蓝创作物科学有限公司 2025-01-07 CN disclosed
WO-2024254056-A1 MODIFIED RELEASE FILL COMPOSITIONS FOR DOSAGE FORMS AND METHODS OF PREPARATION AND USE THEREOF CATALENT ONTARIO LIMITED (CA) 2024-12-12 WO disclosed
CN-116514743-B Paclitaxel-fatty acid prodrug, self-microemulsion preparation, and preparation methods and applications thereof 沈阳药科大学 2024-11-29 CN disclosed
CN-118304270-A Vitamin D drop and preparation method thereof 青岛双鲸药业股份有限公司 2024-07-09 CN disclosed
CN-118078759-A Cefditoren pivoxil granule pharmaceutical composition and preparation method thereof 凌晟(武汉)生物医药技术有限公司 2024-05-28 CN disclosed
US-11969496-B2 Non-greasy personal care compositions COLGATE-PALMOLIVE COMPANY (US) 2024-04-30 US disclosed
CN-117297174-A Filter stick capable of automatically changing taste and preparation method thereof 四川三联新材料有限公司 2023-12-29 CN disclosed
US-11793754-B1 Sodium hypochlorite and chlorhexidine based nanoemulsions and a method of preparation thereof KING ABDULAZIZ UNIVERSITY (SA) 2023-10-24 US disclosed
CN-116898831-A External agent composition containing S-flurbiprofen 江苏恒瑞医药股份有限公司 2023-10-20 CN disclosed
WO-2023187831-A1 A NANO IN MICRO FORMULATION AND PROCESS THEREOF AMRITA VISHWA VIDYAPEETHAM (IN) 2023-10-05 WO disclosed
CN-116514743-A Paclitaxel-fatty acid prodrug, self-microemulsion preparation, and preparation methods and applications thereof 沈阳药科大学 2023-08-01 CN disclosed
US-20220362135-A1 Non-Greasy Personal Care Compositions COLGATE-PALMOLIVE COMPANY (US) 2022-11-17 US disclosed
US-11433018-B2 Non-greasy personal care compositions COLGATE-PALMOLIVE COMPANY (US) 2022-09-06 US disclosed
US-11370996-B2 Compositions including keto-ester compounds and methods of using the same FOURTH PRINCIPLE, LLC (US) 2022-06-28 US disclosed
CN-114591232-A Long-acting control agent for ectoparasites of animals 三井化学AGRO株式会社 2022-06-07 CN disclosed
CN-111132549-B Long-acting control agent for ectoparasites of animals 三井化学AGRO株式会社 2022-04-12 CN disclosed
EP-3179979-B1 NON-GREASY PERSONAL CARE COMPOSITIONS COLGATE PALMOLIVE CO (US) 2021-04-21 EP disclosed
US-20200377823-A1 COMPOSITIONS INCLUDING KETO-ESTER COMPOUNDS AND METHODS OF USING THE SAME TALK ABOUT IT SOLUTIONS 2020-12-03 US disclosed
EP-2525827-B1 PHARMACEUTICAL FORMULATIONS OF LORATADINE FOR ENCAPSULATION AND COMBINATIONS THEREOF CATALENT ONTARIO LTD (CA) 2020-11-18 EP disclosed
EP-3728487-A2 COMPOSITIONS INCLUDING KETO-ESTER COMPOUNDS AND METHODS OF USING THE SAME Fourth Principle, LLC. (US) 2020-10-28 EP disclosed
WO-2020142273-A1 COMPOSITIONS AND METHODS FOR REMOVING COATINGS FROM SURFACES FOURTH PRINCIPLE, LLC (US) 2020-07-09 WO disclosed
EP-3653204-A1 PHARMACEUTICAL FORMULATIONS OF LORATADINE FOR ENCAPSULATION AND COMBINATIONS THEREOF Catalent Ontario Limited (CA) 2020-05-20 EP disclosed
CN-111132549-A Long-acting control agent for ectoparasites of animals 三井化学AGRO株式会社 2020-05-08 CN disclosed
US-20200030223-A1 Non-Greasy Personal Care Compositions COLGATE-PALMOLIVE COMPANY (US) 2020-01-30 US disclosed
US-20190350821-A1 SURFACTANT-FREE EMULSION COMPOSITION GREENVINES BIOTECH CO., LTD. (TW) 2019-11-21 US disclosed
US-10470999-B2 Non-greasy personal care compositions COLGATE-PALMOLIVE COMPANY (US) 2019-11-12 US disclosed
US-10470998-B2 Non-greasy personal care compositions COLGATE-PALMOLIVE COMPANY (US) 2019-11-12 US disclosed
EP-3185845-B1 NON-GREASY PERSONAL CARE COMPOSITIONS COLGATE PALMOLIVE CO (US) 2019-03-27 EP disclosed
US-20170326092-A1 ORAL PHARMACEUTICAL COMPOSITION OF ISOTRETINOIN SUN PHARMACEUTICAL INDUSTRIES LIMITED (IN) 2017-11-16 US disclosed
US-20170252288-A1 Non-Greasy Personal Care Compositions COLGATE-PALMOLIVE COMPANY (US) 2017-09-07 US disclosed
US-20170246104-A1 Non-Greasy Personal Care Compositions COLGATE-PALMOLIVE COMPANY (US) 2017-08-31 US disclosed
EP-3185845-A1 NON-GREASY PERSONAL CARE COMPOSITIONS Colgate-Palmolive Company (US) 2017-07-05 EP disclosed
EP-3179979-A1 NON-GREASY PERSONAL CARE COMPOSITIONS Colgate-Palmolive Company (US) 2017-06-21 EP disclosed
EP-3148645-A1 ORAL PHARMACEUTICAL COMPOSITION OF ISOTRETINOIN Sun Pharmaceutical Industries Ltd (IN) 2017-04-05 EP disclosed
WO-2016048425-A1 NON-GREASY PERSONAL CARE COMPOSITIONS COLGATE-PALMOLIVE COMPANY (US) 2016-03-31 WO disclosed
WO-2016048274-A1 NON-GREASY PERSONAL CARE COMPOSITIONS COLGATE-PALMOLIVE COMPANY (US) 2016-03-31 WO disclosed
US-20160081965-A1 ORAL PHARMACEUTICAL COMPOSITION OF ISOTRETINOIN SUN PHARMACEUTICAL INDUSTRIES LIMITED (IN) 2016-03-24 US disclosed
WO-2015186039-A1 ORAL PHARMACEUTICAL COMPOSITION OF ISOTRETINOIN SUN PHARMACEUTICAL INDUSTRIES LIMITED (IN) 2015-12-10 WO disclosed
EP-2877178-A1 PHARMACEUTICAL COMPOSITION COMPRISING DIAMORPHINE FOR INTRANASAL ADMINISTRATION Wockhardt Limited (IN) 2015-06-03 EP disclosed
WO-2015059466-A1 PHARMACEUTICAL COMPOSITIONS COMPRISING EFAVIRENZ CIPLA LIMITED (IN) 2015-04-30 WO disclosed
WO-2014016653-A1 PHARMACEUTICAL COMPOSITION COMPRISING DIAMORPHINE FOR INTRANASAL ADMINISTRATION WOCKHARDT LIMITED (IN) 2014-01-30 WO disclosed
WO-2013088274-A1 ANHYDROUS AMORPHOUS AZITHROMYCIN COMPOSITION FREE OF AZITHROMYCIN DIHYDRATE WOCKHARDT LIMITED (IN) 2013-06-20 WO disclosed
WO-2013008083-A1 PHARMACEUTICAL COMPOSITION FOR ENHANCING ANTICANCER EFFICACY OF TAMOXIFEN NATIONAL INSTITUTE OF PHARMACEUTICAL EDUCATION AND RESEARCH (NIPER) (IN) 2013-01-17 WO disclosed
EP-2544887-A1 A DEVICE FOR THE MANUFACTURE OF A DOSAGE FORM WITH A HOLE AND METHOD OF MANUFACTURE Wockhardt Limited (IN) 2013-01-16 EP disclosed
EP-2542243-A2 MODIFIED RELEASE DOSAGE FORM Wockhardt Limited (IN) 2013-01-09 EP disclosed
US-20120301544-A1 PHARMACEUTICAL FORMULATIONS OF LORATADINE FOR ENCAPSULATION AND COMBINATIONS THEREOF ACCUCAPS INDUSTRIES LIMITED (CA) 2012-11-29 US disclosed
EP-2521537-A2 PHARMACEUTICAL COMPOSITION FOR MODIFIED DELIVERY OF ACTIVES Wockhardt Limited (IN) 2012-11-14 EP disclosed
WO-2011110989-A1 A DEVICE FOR THE MANUFACTURE OF A DOSAGE FORM WITH A HOLE AND METHOD OF MANUFACTURE WOCKHARDT LIMITED (IN) 2011-09-15 WO disclosed
WO-2011107944-A2 MODIFIED RELEASE DOSAGE FORM WOCKHARDT LIMITED (IN) 2011-09-09 WO disclosed
WO-2011088550-A1 PHARMACEUTICAL FORMULATIONS OF LORATADINE FOR ENCAPSULATION AND COMBINATIONS THEREOF ACCUCAPS INDUSTRIES LIMITED (CA) 2011-07-28 WO disclosed
WO-2011080716-A2 PHARMACEUTICAL COMPOSITION FOR MODIFIED DELIVERY OF ACTIVES WOCKHARDT LIMITED (IN) 2011-07-07 WO disclosed
WO-2011004395-A1 MICROEMULSION FORMULATION FOR BIOLOGICALS INTAS BIOPHARMACEUTICALS LIMITED (IN) 2011-01-13 WO disclosed
US-20080118490-A1 Combined use of triglycerides containing medium chain fatty acids and exogenous lipolytic enzymes as feed supplements VITAMEX,N.V. (BE) 2008-05-22 US disclosed
EP-0995430-A2 Use of diacylolycerols for enhancing the barrier function of the skin Beiersdorf Aktiengesellschaft (DE) 2000-04-26 EP disclosed
EP-0655907-B1 USE OF DIACYLOLYCEROLS FOR INCREASING THE MELANIN CONTENT IN MELANOCYTES UNIV BOSTON (US) 1999-04-28 EP disclosed
US-5750091-A Methods for increasing melanin content in melanocytes using diacylglycerols and uses thereof THE TRUSTEES OF BOSTON UNIVERSITY (US) 1998-05-12 US disclosed
US-5700450-A Methods for enhancing melanin synthesis in melanocytes using diacyglycerols and uses thereof THE TRUSTEES OF BOSTON UNIVERSITY (US) 1997-12-23 US disclosed
EP-0542108-B1 Stabilizers for plastic materials CIBA GEIGY AG (CH) 1997-09-24 EP disclosed
JP-H08245830-A STABILIZER FOR PLASTIC MATERIAL F HOFFMANN LA ROCHE AG 1996-09-24 JP disclosed
EP-0730001-A1 Stabilizers for plastic materials F. HOFFMANN-LA ROCHE AG (CH) 1996-09-04 EP disclosed
US-5352440-A Methods for increasing melanin content in melanocytes using diacylglycerols and uses thereof TRUSTEES OF BOSTON UNIVERSITY (US) 1994-10-04 US disclosed
US-5308549-A OF ALPHA-TOCOPHEROL, GLYCERIN, POLYOXYETHYLENE GLYCOL AND GLYCERYL MONOCAPRYLATE-CAPRATE HOFFMANN-LA ROCHE INC. (US) 1994-05-03 US disclosed
EP-0566718-A1 STABILIZERS FOR PLASTIC MATERIALS Ciba SC Holding AG (CH) 1993-10-27 EP disclosed
WO-1993010175-A1 STABILIZERS FOR PLASTIC MATERIALS F. HOFFMANN-LA ROCHE AG (CH) 1993-05-27 WO disclosed
EP-0542108-A2 Stabilizers for plastic materials F. HOFFMANN-LA ROCHE AG (CH) 1993-05-19 EP disclosed
EP-0542108-A2 Stabilizers for plastic materials F. HOFFMANN-LA ROCHE AG (CH) 1993-05-19 EP disclosed
EP-0542108-A2 Stabilizers for plastic materials F. HOFFMANN-LA ROCHE AG (CH) 1993-05-19 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20260042933-A1 Formulation For Simultaneous Rejuvenation And Protection Of The Interior Fibers And Exterior Surfaces Of Wood PPARA, ELOVL1, ELOVL3 PRKCA 2717/4885PRKCE 1880/4885PRKCQ 3766/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.