SCHEMBL10048196

SCHEMBL10048196

C=Cc1cnc(N(C)C(=O)OC(C)(C)C)c(Oc2ccc(C)cc2)n1

nearest known ligand 0.35

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
LIPE Q05469 3/20 0.35
CYP1A2 P05177 1/20 0.32
CYP3A4 P08684 1/20 0.32
CYP2C9 P11712 1/20 0.32
CYP2C19 P33261 1/20 0.32
MEN1 O00255 2/20 0.32
KMT2A Q03164 2/20 0.32
ALDH1A1 P00352 3/20 0.31
NPC1 O15118 1/20 0.31
HPGD P15428 1/20 0.31
HTT P42858 1/20 0.31
RAB9A P51151 1/20 0.31
ATM Q13315 1/20 0.31
PAX8 Q06710 1/20 0.31
KDM4E B2RXH2 1/20 0.30
LMNA P02545 1/20 0.30
MAPT P10636 1/20 0.30
HSD17B1 P14061 1/20 0.30
HSD17B2 P37059 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10048194 0.73 KMT2A (0.34) LIPECYP1A2CYP3A4CYP2C9CYP2C19
SCHEMBL17340121 0.73 KMT2A (0.34) LIPECYP1A2CYP3A4CYP2C9CYP2C19
SCHEMBL15215741 0.72 ALDH1A1 (0.39) CYP1A2CYP3A4CYP2C9CYP2C19MEN1
SCHEMBL25227083 0.66 NPSR1 (0.33) ALDH1A1
SCHEMBL14384381 0.65 PAX8 (0.50) LIPECYP1A2CYP3A4CYP2C9CYP2C19
SCHEMBL20037705 0.65 TTK (0.39) LIPEMEN1KMT2AALDH1A1NPC1
SCHEMBL10325135 0.64 NPSR1 (0.33) ALDH1A1
SCHEMBL6177591 0.63 TTK (0.35) ALDH1A1NPC1RAB9APAX8KDM4E
SCHEMBL27804098 0.63 HSD17B1 (0.40) LIPEALDH1A1HTTLMNAMAPT
SCHEMBL19219152 0.62 STK17B (0.38) ALDH1A1PAX8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012020742-A1 NOVEL HETEROCYCLIC DERIVATIVES AND PHARMACEUTICAL COMPOSITION CONTAINING SAME 塩野義製薬株式会社 (JP) 2012-02-16 WO disclosed