SCHEMBL10049030

SCHEMBL10049030

N#Cc1ccc(-c2ccc(N)cc2F)c2c1C(=O)NC2

nearest known ligand 0.46

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
BTK Q06187 9/20 0.46
TYK2 P29597 9/20 0.36
JAK2 O60674 8/20 0.36
KDM1A O60341 1/20 0.36
KDR P35968 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12469593 0.95 BTK (0.44) BTKTYK2JAK2KDM1AKDR
SCHEMBL1334382 0.77 KDR (0.54) KDR
SCHEMBL12469189 0.77 BTK (0.46) BTKKDR
SCHEMBL10048588 0.75 BTK (0.44) BTKKDR
SCHEMBL12469765 0.75 AURKA (0.40) BTKKDR
SCHEMBL12469516 0.75 GRM2 (0.40) BTKKDR
SCHEMBL10049027 0.74 PARP1 (0.35) BTKTYK2JAK2KDR
SCHEMBL12469667 0.73 BTK (0.43) BTK
SCHEMBL12469427 0.73 BTK (0.67) BTKKDR
SCHEMBL12469609 0.72 BTK (0.39) BTKKDR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012047017-A2 2,3-DIHYDRO-ISOINDOL-1-ONE DERIVATIVE AND A COMPOSITION COMPRISING THE SAME 크리스탈지노믹스(주) (KR) 2012-04-12 WO disclosed