SCHEMBL12469765

SCHEMBL12469765

NC(=O)c1ccc(-c2ccc(N)cc2F)c2c1C(=O)NC2.Nc1ccc(F)cc1

nearest known ligand 0.40

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
AURKA O14965 1/20 0.40
BTK Q06187 13/20 0.40
KDR P35968 2/20 0.36
FLT3 P36888 1/20 0.36
GRM2 Q14416 1/20 0.35
GRM5 P41594 1/20 0.33
IKBKB O14920 1/20 0.33
CHUK O15111 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12469562 0.87 BTK (0.42) BTKKDRFLT3GRM2IKBKB
SCHEMBL12469505 0.85 BTK (0.41) BTKKDRFLT3
SCHEMBL12469629 0.85 KDR (0.41) AURKABTKKDRGRM2IKBKB
SCHEMBL12469508 0.84 BTK (0.40) BTKKDRFLT3
SCHEMBL12469481 0.84 ALOX5 (0.40) BTKKDRFLT3
SCHEMBL12469512 0.84 CRBN (0.41) BTK
SCHEMBL12469573 0.84 ALPL (0.40) BTKKDRFLT3
SCHEMBL1292654 0.83 BTK (0.57) AURKABTKKDRFLT3
SCHEMBL10048588 0.82 BTK (0.44) BTKKDRFLT3
SCHEMBL12469516 0.82 GRM2 (0.40) BTKKDRFLT3GRM2GRM5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012047017-A2 2,3-DIHYDRO-ISOINDOL-1-ONE DERIVATIVE AND A COMPOSITION COMPRISING THE SAME 크리스탈지노믹스(주) (KR) 2012-04-12 WO disclosed