SCHEMBL12469593

SCHEMBL12469593

N#Cc1ccc(-c2ccc(N)cc2F)c2c1C(=O)NC2.Nc1ccc(F)cc1

nearest known ligand 0.44

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
BTK Q06187 8/20 0.44
GRM5 P41594 1/20 0.36
GRM2 Q14416 1/20 0.36
MEN1 O00255 1/20 0.36
KMT2A Q03164 1/20 0.36
JAK2 O60674 5/20 0.34
TYK2 P29597 5/20 0.34
KDM1A O60341 1/20 0.34
RIPK3 Q9Y572 1/20 0.34
KDR P35968 1/20 0.33
PDE3B Q13370 1/20 0.32
PDE3A Q14432 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10049030 0.95 BTK (0.46) BTKJAK2TYK2KDM1AKDR
SCHEMBL12469516 0.81 GRM2 (0.40) BTKGRM5GRM2KDRPDE3B
SCHEMBL12469765 0.81 AURKA (0.40) BTKGRM5GRM2KDR
SCHEMBL12469667 0.79 BTK (0.43) BTKGRM2PDE3BPDE3A
SCHEMBL12469271 0.78 NISCH (0.43) BTKGRM2
SCHEMBL12469609 0.78 BTK (0.39) BTKGRM2KDRPDE3BPDE3A
SCHEMBL12469700 0.77 BTK (0.40) BTKGRM5GRM2KDRPDE3B
SCHEMBL12469562 0.77 BTK (0.42) BTKGRM2KDR
SCHEMBL12469647 0.77 BTK (0.38) BTKGRM5GRM2PDE3BPDE3A
SCHEMBL12469863 0.76 BTK (0.42) BTKGRM2TYK2PDE3BPDE3A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012047017-A2 2,3-DIHYDRO-ISOINDOL-1-ONE DERIVATIVE AND A COMPOSITION COMPRISING THE SAME 크리스탈지노믹스(주) (KR) 2012-04-12 WO disclosed