SCHEMBL10051168

SCHEMBL10051168

COc1cc(C)c(-c2c(OC)cc(C)cc2OC)c(OC)c1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ACHE P22303 3/20 0.46
ALDH1A1 P00352 3/20 0.46
CYP1A2 P05177 1/20 0.46
CYP3A4 P08684 1/20 0.46
PTPN1 P18031 2/20 0.45
NQO2 P16083 2/20 0.42
CA12 O43570 1/20 0.40
CA1 P00915 1/20 0.40
CA2 P00918 1/20 0.40
CA7 P43166 1/20 0.40
CA9 Q16790 1/20 0.40
CA14 Q9ULX7 1/20 0.40
ELANE P08246 1/20 0.40
CYP19A1 P11511 1/20 0.40
KDM4E B2RXH2 1/20 0.39
LMNA P02545 1/20 0.39
GAA P10253 1/20 0.39
HPGD P15428 1/20 0.39
HSD17B10 Q99714 1/20 0.39
TDP1 Q9NUW8 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15120000 0.91 ALDH1A1 (0.52) ACHEALDH1A1CYP1A2CYP3A4NQO2
Difucol Hexamethyl Ether SCHEMBL505203 0.82 CYP1A2 (0.60) ACHEALDH1A1CYP1A2CYP3A4NQO2
SCHEMBL26328948 0.82 ALDH1A1 (0.44) ACHEALDH1A1CYP1A2CYP3A4NQO2
SCHEMBL15119996 0.80 ALDH1A1 (0.43) ACHEALDH1A1CYP1A2CYP3A4NQO2
SCHEMBL12326164 0.77 ALDH1A1 (0.59) ACHEALDH1A1CYP1A2CYP3A4PTPN1
SCHEMBL17930308 0.75 MAPT (0.49) ALDH1A1CYP1A2CYP3A4CA12CA1
SCHEMBL16624733 0.75 ACHE (0.42) ACHEALDH1A1CYP1A2CYP3A4PTPN1
SCHEMBL26201033 0.73 ACHE (0.45) ACHEALDH1A1CRHR1
SCHEMBL15488875 0.73 ACHE (0.41) ACHEALDH1A1CYP1A2CYP3A4PTPN1
SCHEMBL890469 0.73 ERN1 (0.46) ACHEALDH1A1CYP1A2CYP3A4PTPN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9273021-B2 Dibenzofuran derivatives as inhibitors of fructose 1,6-bisphosphatase and methods of use thereof TRUSTEES OF BOSTON COLLEGE (US) 2016-03-01 US disclosed
US-20120028892-A1 INHIBITORS OF FRUCTOSE 1,6-BISPHOSPHATASE AND METHODS OF USE THEREOF TRUSTEES OF BOSTON COLLEGE (US) 2012-02-02 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20120028892-A1 INHIBITORS OF FRUCTOSE 1,6-BISPHOSPHATASE AND METHODS OF USE THEREOF FBP1, SLC5A1, ALDOA ACHE 1565/4885ALDH1A1 279/4885CYP1A2 429/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.