SCHEMBL10055700

SCHEMBL10055700

Cc1ccc(Cn2c(Cc3ccccc3)nc(=O)[nH]c2=O)cc1

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 4/20 0.60
KMT2A Q03164 4/20 0.60
TP53 P04637 4/20 0.60
HTT P42858 3/20 0.60
LMNA P02545 2/20 0.60
SMN1; SMN2 Q16637 2/20 0.60
MAPT P10636 1/20 0.60
ADORA3 P0DMS8 1/20 0.49
HPGD P15428 4/20 0.47
KDM4E B2RXH2 3/20 0.47
PSMD14 O00487 1/20 0.47
TSHR P16473 1/20 0.47
ALDH1A1 P00352 2/20 0.46
RGS4 P49798 1/20 0.46
RGS8 P57771 1/20 0.46
PDE5A O76074 1/20 0.45
TLR7 Q9NYK1 3/20 0.45
NPSR1 Q6W5P4 1/20 0.45
GAA P10253 1/20 0.44
P2RX3 P56373 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10048444 0.73 P2RX3 (0.56) MEN1KMT2ATP53HTTLMNA
SCHEMBL6502344 0.72 ALDH1A1 (0.51) LMNASMN1; SMN2MAPTHPGDKDM4E
SCHEMBL26790950 0.71 BRAF (0.61) MEN1KMT2AHTTSMN1; SMN2HPGD
SCHEMBL11721250 0.71 P2RX4 (0.49) MEN1KMT2ATP53LMNASMN1; SMN2
SCHEMBL12045850 0.70 P2RX3 (0.52) MEN1KMT2AHTTLMNASMN1; SMN2
SCHEMBL9527922 0.69 DAO (0.46) MEN1KMT2ATP53LMNAMDM2
SCHEMBL97080 0.69 LMNA (0.55) MEN1KMT2ATP53HTTLMNA
SCHEMBL29989784 0.69 LMNA (0.53) HTTLMNATLR7P2RX3
SCHEMBL10048214 0.69 P2RX3 (0.77) MEN1KMT2ATP53HTTLMNA
SCHEMBL19291210 0.68 HPGD (0.80) MEN1KMT2ATP53HTTLMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9718790-B2 Triazine derivative and pharmaceutical composition having an analgesic activity comprising the same SHIONOGI & CO., LTD. (JP) 2017-08-01 US disclosed
US-9718790-B2 Triazine derivative and pharmaceutical composition having an analgesic activity comprising the same SHIONOGI & CO., LTD. (JP) 2017-08-01 US disclosed
EP-2604595-B1 TRIAZINE DERIVATIVE AND PHARMACEUTICAL COMPOUND THAT CONTAINS SAME AND EXHIBITS ANALGESIC ACTIVITY SHIONOGI & CO (JP) 2016-03-16 EP disclosed
WO-2012020749-A1 TRIAZINE DERIVATIVE AND PHARMACEUTICAL COMPOUND THAT CONTAINS SAME AND EXHIBITS ANALGESIC ACTIVITY 塩野義製薬株式会社 (JP) 2012-02-16 WO disclosed