SCHEMBL10057071

SCHEMBL10057071

C[C@@H](CN(C(N)=O)C(=O)NCc1ccc(Cl)cn1)C(=O)O

nearest known ligand 0.37

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
WDR5 P61964 4/20 0.37
MAOB P27338 1/20 0.37
MAPK1 P28482 2/20 0.36
L3MBTL1 Q9Y468 1/20 0.36
KCNH2 Q12809 1/20 0.35
HRH3 Q9Y5N1 1/20 0.35
P2RX3 P56373 2/20 0.34
RORC P51449 1/20 0.33
CYP1A2 P05177 1/20 0.33
CYP2D6 P10635 1/20 0.33
MAPT P10636 1/20 0.33
TSHR P16473 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
KMO O15229 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10055489 0.82 CYP2C9 (0.50) L3MBTL1TSHRSMN1; SMN2
SCHEMBL10055215 0.73 SMN1; SMN2 (0.46) SMN1; SMN2
SCHEMBL10056387 0.71 CARM1 (0.47) SMN1; SMN2
SCHEMBL10055319 0.71 CYP2C9 (0.48) MAPK1L3MBTL1CYP1A2CYP2D6MAPT
SCHEMBL30791568 0.70 PTK2 (0.53) WDR5MAOBMAPK1L3MBTL1
SCHEMBL10056326 0.69 ALDH1A1 (0.37) MAPK1P2RX3MAPTTSHRSMN1; SMN2
SCHEMBL15044016 0.67
SCHEMBL18080787 0.66 L3MBTL1 (0.45) MAOBMAPK1L3MBTL1P2RX3MAPT
Hydrochloric Acid SCHEMBL25217806 0.65 CYP1A2 (0.46) CYP1A2KMO
SCHEMBL26459530 0.64 WDR5 (0.42) WDR5MAOBMAPK1L3MBTL1SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012020749-A1 TRIAZINE DERIVATIVE AND PHARMACEUTICAL COMPOUND THAT CONTAINS SAME AND EXHIBITS ANALGESIC ACTIVITY 塩野義製薬株式会社 (JP) 2012-02-16 WO disclosed