SCHEMBL10059752

SCHEMBL10059752

Cc1cc(OS(=O)(=O)C(F)(F)F)c(C)cc1N

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 1/20 0.39
TSHR P16473 1/20 0.39
MAPK1 P28482 1/20 0.39
POLB P06746 1/20 0.34
GAA P10253 1/20 0.34
GFER P55789 1/20 0.34
ALDH1A1 P00352 2/20 0.33
AR P10275 1/20 0.33
STS P08842 1/20 0.33
CA1 P00915 2/20 0.32
CA2 P00918 2/20 0.32
DRD2 P14416 1/20 0.32
DRD1 P21728 1/20 0.32
DRD4 P21917 1/20 0.32
DRD5 P21918 1/20 0.32
DRD3 P35462 1/20 0.32
HTR1A P08908 1/20 0.31
HTR1D P28221 1/20 0.31
HTR1B P28222 1/20 0.31
ADORA2A P29274 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6938167 0.85 DRD2 (0.34) STSCA1CA2DRD2DRD1
SCHEMBL17864633 0.82 MEN1 (0.41) TSHRMAPK1POLBGAAALDH1A1
SCHEMBL14240535 0.81 DRD2 (0.38) CA1CA2DRD2DRD1DRD4
SCHEMBL26601703 0.78 ALDH1A1 (0.31) ALDH1A1DRD2DRD1DRD4DRD5
SCHEMBL18179589 0.76 EPAS1 (0.38) TSHRMAPK1POLBCA1CA2
SCHEMBL5156307 0.75 AR (0.50) ARSTSDRD2DRD1DRD4
SCHEMBL6139736 0.75 RAB9A (0.40) POLBALDH1A1STSCA1CA2
Hydrogen Sulfide SCHEMBL15796096 0.74 ESR2 (0.33) CA1CA2DRD2DRD1DRD4
SCHEMBL6942043 0.74 CA1 (0.44) TSHRGAAALDH1A1CA1CA2
SCHEMBL31195498 0.74 CA1 (0.44) GAAALDH1A1STSCA1CA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012086735-A1 CONDENSED HETEROCYCLIC COMPOUND 大正製薬株式会社 (JP) 2012-06-28 WO disclosed