SCHEMBL10065075

SCHEMBL10065075

CC(C)n1cc(-c2ccc(NC(=O)c3cc4c(s3)N=CCC4)cc2)cc1C(=O)NC1CC1

nearest known ligand 0.34

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LRRK2 Q5S007 3/20 0.34
MAPT P10636 6/20 0.34
NPC1 O15118 4/20 0.34
ALDH1A1 P00352 3/20 0.34
RAB9A P51151 3/20 0.34
KDM4E B2RXH2 3/20 0.34
LMNA P02545 2/20 0.34
NFKB1 P19838 1/20 0.34
NFKB2 Q00653 1/20 0.34
RELA Q04206 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
MEN1 O00255 1/20 0.34
KMT2A Q03164 1/20 0.34
DGAT1 O75907 3/20 0.34
ABL1 P00519 1/20 0.34
PRNP P04156 1/20 0.33
MAPK1 P28482 2/20 0.33
TP53 P04637 1/20 0.33
PDE7A Q13946 2/20 0.32
NAMPT P43490 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL876773 0.72 LRRK2 (0.42) LRRK2NPC1RAB9AKDM4ESMN1; SMN2
SCHEMBL876507 0.69 MAPT (0.46) LRRK2MAPTALDH1A1KMT2A
SCHEMBL876612 0.62 CHRNA7 (0.46) NPC1RAB9AKMT2ANAMPTMAPK14
SCHEMBL10225025 0.57 LRRK2 (0.85) LRRK2
SCHEMBL874150 0.54 HDAC6 (0.48) KDM4EMAPK14
SCHEMBL16708659 0.54 THRB (0.47) MAPTALDH1A1KDM4ELMNAMEN1
SCHEMBL20365093 0.54 BRD4 (0.52) MAPTNPC1RAB9ASMN1; SMN2MEN1
SCHEMBL15723817 0.54 BRD4 (0.50) NPC1ALDH1A1RAB9AKDM4ESMN1; SMN2
SCHEMBL14009108 0.53 SMYD3 (0.53) MAPTNPC1ALDH1A1RAB9AKDM4E
SCHEMBL882712 0.53 HDAC6 (0.47) KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012038905-A1 THIENOPYRIDINE NICOTINAMIDE DERIVATIVES, PREPARATION THEREOF AND THERAPEUTIC USE THEREOF SANOFI (FR) 2012-03-29 WO disclosed