SCHEMBL10068677

SCHEMBL10068677

Cc1ccc(N(c2ccc(C#N)cc2)c2cc(C)c3ccc4c(N(c5ccc(C)cc5)c5ccc(C#N)cc5)cc(C)c5ccc2c3c54)cc1

nearest known ligand 0.47

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
CYP2A6 P11509 2/20 0.47
ALDH1A1 P00352 1/20 0.47
HCRTR2 O43614 1/20 0.36
GRM2 Q14416 1/20 0.34
RORC P51449 4/20 0.33
AR P10275 1/20 0.33
NOS3 P29474 1/20 0.32
NOS1 P29475 1/20 0.32
MAPKAPK2 P49137 1/20 0.32
BCHE P06276 1/20 0.31
ACHE P22303 1/20 0.31
CHEK1 O14757 1/20 0.31
KDM1A O60341 3/20 0.31
CSNK1A1 P48729 1/20 0.30
CSNK1D P48730 1/20 0.30
GSK3B P49841 1/20 0.30
CSNK1G2 P78368 1/20 0.30
IDO1 P14902 1/20 0.30
IDH1 O75874 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10069240 0.95 ALDH1A1 (0.38) CYP2A6ALDH1A1HCRTR2GRM2NOS3
SCHEMBL10118867 0.95 ALDH1A1 (0.42) CYP2A6ALDH1A1HCRTR2GRM2RORC
SCHEMBL19505954 0.94 CYP2A6 (0.37) CYP2A6ALDH1A1GRM2NOS3NOS1
SCHEMBL10069121 0.92 CYP2A6 (0.37) CYP2A6ALDH1A1HCRTR2GRM2NOS3
SCHEMBL10038682 0.90 ALDH1A1 (0.38) CYP2A6ALDH1A1HCRTR2
SCHEMBL10068689 0.90 CRHBP (0.37) CYP2A6ALDH1A1RORCARNOS3
SCHEMBL12768343 0.87 ALDH1A1 (0.37) ALDH1A1ACHE
SCHEMBL10069123 0.87 CYP2A6 (0.51) CYP2A6ALDH1A1NOS3NOS1ACHE
SCHEMBL10068680 0.86 S1PR1 (0.36) CYP2A6ALDH1A1NOS3NOS1
SCHEMBL17715238 0.86 NOS3 (0.32) CYP2A6ALDH1A1NOS3NOS1CHEK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9923146-B2 Aromatic amine derivative and organic electroluminescent element using same IDEMITSU KOSAN CO., LTD. (JP) 2018-03-20 US disclosed
US-20170309822-A1 AROMATIC AMINE DERIVATIVE AND ORGANIC ELECTROLUMINESCENT ELEMENT USING SAME IDEMITSU KOSAN CO., LTD. (JP) 2017-10-26 US disclosed
US-20160181527-A1 AROMATIC AMINE DERIVATIVE AND ORGANIC ELECTROLUMINESCENT ELEMENT USING SAME IDEMITSU KOSAN CO., LTD. (JP) 2016-06-23 US disclosed
US-9331285-B2 Aromatic amine derivative and organic electroluminescent element using same IDEMITSU KOSAN CO., LTD. (JP) 2016-05-03 US disclosed
US-20120013244-A1 ORGANIC LUMINESCENT MEDIUM IDEMITSU KOSAN CO., LTD. 2012-01-19 US disclosed
US-20110297923-A1 Aromatic amine derivative and organic electroluminescent element using same IDEMITSU KOSAN CO., LTD. 2011-12-08 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20120013244-A1 ORGANIC LUMINESCENT MEDIUM ANXA1, ANXA11, GLB1 CYP2A6 1167/4885ALDH1A1 61/4885HCRTR2 4356/4885
US-20170309822-A1 AROMATIC AMINE DERIVATIVE AND ORGANIC ELECTROLUMINESCENT ELEMENT USING SAME H1-4, H1-2, H1-0 CYP2A6 3351/4885ALDH1A1 672/4885HCRTR2 1268/4885
US-20110297923-A1 Aromatic amine derivative and organic electroluminescent element using same H1-4, H1-2, H1-0 CYP2A6 3351/4885ALDH1A1 672/4885HCRTR2 1268/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.