SCHEMBL10069630

SCHEMBL10069630

CCc1c(-c2ccc3ccccc3c2)n(COCc2ccccc2)c(=O)n(O)c1=O

nearest known ligand 0.38

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.38
KDM5B Q9UGL1 1/20 0.33
ALOX5 P09917 1/20 0.33
MAPK14 Q16539 1/20 0.33
POLB P06746 1/20 0.33
RECQL P46063 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
CNOT7 Q9UIV1 1/20 0.32
NPC1 O15118 1/20 0.32
RAB9A P51151 1/20 0.32
ERCC5 P28715 1/20 0.32
FEN1 P39748 1/20 0.32
ESR1 P03372 1/20 0.32
USP2 O75604 1/20 0.32
MAPK1 P28482 1/20 0.32
KDM4E B2RXH2 1/20 0.32
CYSLTR1 Q9Y271 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10069632 0.88 ALDH1A1 (0.43) ALDH1A1KDM5BMAPK14POLBRECQL
SCHEMBL10069623 0.86 ALDH1A1 (0.42) ALDH1A1MAPK14POLBRECQLSMN1; SMN2
SCHEMBL10069613 0.85 ALDH1A1 (0.40) ALDH1A1POLBRECQLSMN1; SMN2NPC1
SCHEMBL10069591 0.85 ESR1 (0.35) ALDH1A1KDM5BALOX5ERCC5FEN1
SCHEMBL10069625 0.85 ALDH1A1 (0.41) ALDH1A1KDM5BMAPK14POLBRECQL
SCHEMBL10069621 0.85 ALDH1A1 (0.39) ALDH1A1MAPK14SMN1; SMN2NPC1RAB9A
SCHEMBL1287915 0.85 ALDH1A1 (0.39) ALDH1A1MAPK14POLBRECQLSMN1; SMN2
SCHEMBL10069600 0.82 AR (0.42) ALDH1A1POLBNPC1RAB9AKDM4E
SCHEMBL10069617 0.81 ALDH1A1 (0.35) ALDH1A1MAPK14POLBCNOT7ERCC5
SCHEMBL1687638 0.79 ADORA2A (0.36) ALDH1A1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012047993-A2 N-HYDROXYPYRIMIDINE-2,4-DIONES AS INHIBITORS OF HIV AND HCV REGENTS OF THE UNIVERSITY OF MINNESOTA (US) 2012-04-12 WO disclosed