SCHEMBL10069591

SCHEMBL10069591

CC(C)c1c(-c2ccc3ccccc3c2)n(COCc2ccccc2)c(=O)n(O)c1=O

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 1/20 0.35
ALDH1A1 P00352 1/20 0.35
CASR P41180 1/20 0.34
ALOX5 P09917 1/20 0.33
LMNA P02545 1/20 0.33
MEN1 O00255 1/20 0.33
KMT2A Q03164 1/20 0.33
IDH1 O75874 1/20 0.33
KDM5B Q9UGL1 1/20 0.32
MAPK1 P28482 2/20 0.32
ERCC5 P28715 2/20 0.32
FEN1 P39748 2/20 0.32
USP2 O75604 1/20 0.32
CTSL P07711 1/20 0.32
CTSB P07858 1/20 0.32
CTSS P25774 1/20 0.32
CYP1A2 P05177 1/20 0.32
PDE10A Q9Y233 1/20 0.32
CYSLTR1 Q9Y271 1/20 0.32
MAOB P27338 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10069597 0.92 ANO1 (0.36) ESR1LMNAKDM5BPDE10A
SCHEMBL10069590 0.89 ALDH1A1 (0.39) ALDH1A1LMNAIDH1KDM5BMAPK1
SCHEMBL10069606 0.87 ALDH1A1 (0.37) ALDH1A1CASRLMNAKMT2AIDH1
SCHEMBL10069595 0.86 ALDH1A1 (0.38) ALDH1A1LMNAIDH1MAPK1ERCC5
SCHEMBL10069601 0.86 ALDH1A1 (0.36) ALDH1A1MEN1KMT2AMAPK1ERCC5
SCHEMBL10069594 0.86 MAPT (0.38) ALDH1A1LMNAERCC5FEN1USP2
SCHEMBL10069630 0.85 ALDH1A1 (0.38) ESR1ALDH1A1ALOX5KDM5BMAPK1
SCHEMBL10069592 0.84 MEN1 (0.40) ALDH1A1MEN1KMT2A
SCHEMBL10069620 0.82 MAPK1 (0.36) ALDH1A1CASRMAPK1ERCC5FEN1
SCHEMBL10069611 0.82 L3MBTL1 (0.36) ALDH1A1USP2CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012047993-A2 N-HYDROXYPYRIMIDINE-2,4-DIONES AS INHIBITORS OF HIV AND HCV REGENTS OF THE UNIVERSITY OF MINNESOTA (US) 2012-04-12 WO disclosed