SCHEMBL1287915

SCHEMBL1287915

CCc1c(-c2ccc(F)cc2)n(COCc2ccccc2)c(=O)n(O)c1=O

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.39
SLC34A1 Q06495 1/20 0.36
CYP2C9 P11712 2/20 0.36
CYP2C19 P33261 2/20 0.36
GRM5 P41594 1/20 0.35
MEN1 O00255 2/20 0.35
CYP1A2 P05177 2/20 0.35
CASP1 P29466 2/20 0.35
CASP7 P55210 2/20 0.35
KMT2A Q03164 2/20 0.35
HSD17B10 Q99714 2/20 0.35
MAPK14 Q16539 1/20 0.34
L3MBTL1 Q9Y468 1/20 0.34
AR P10275 1/20 0.34
ASAH1 Q13510 1/20 0.34
POLB P06746 1/20 0.34
RECQL P46063 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
CYP3A4 P08684 1/20 0.34
HPGD P15428 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1687638 0.94 ADORA2A (0.36) ALDH1A1SLC34A1HSD17B10L3MBTL1AR
SCHEMBL10069632 0.92 ALDH1A1 (0.43) ALDH1A1MAPK14POLBRECQLSMN1; SMN2
SCHEMBL10069623 0.90 ALDH1A1 (0.42) ALDH1A1MEN1KMT2AMAPK14AR
SCHEMBL10069621 0.89 ALDH1A1 (0.39) ALDH1A1GRM5CYP1A2KMT2AHSD17B10
SCHEMBL10069600 0.85 AR (0.42) ALDH1A1MEN1KMT2AARPOLB
SCHEMBL10069630 0.85 ALDH1A1 (0.38) ALDH1A1MAPK14POLBRECQLSMN1; SMN2
SCHEMBL10069625 0.85 ALDH1A1 (0.41) ALDH1A1GRM5MAPK14POLBRECQL
SCHEMBL10069601 0.84 ALDH1A1 (0.36) ALDH1A1CYP2C9CYP2C19GRM5MEN1
SCHEMBL10069613 0.83 ALDH1A1 (0.40) ALDH1A1MEN1KMT2AL3MBTL1AR
SCHEMBL1287928 0.82 ALDH1A1 (0.53) ALDH1A1SLC34A1CYP2C9CYP2C19L3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012047993-A2 N-HYDROXYPYRIMIDINE-2,4-DIONES AS INHIBITORS OF HIV AND HCV REGENTS OF THE UNIVERSITY OF MINNESOTA (US) 2012-04-12 WO disclosed
WO-2012047993-A2 N-HYDROXYPYRIMIDINE-2,4-DIONES AS INHIBITORS OF HIV AND HCV REGENTS OF THE UNIVERSITY OF MINNESOTA (US) 2012-04-12 WO disclosed