SCHEMBL10069798

SCHEMBL10069798

COc1ccc(C(=O)C#Cc2ccccc2)cc1

nearest known ligand 0.72

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
APP P05067 1/20 0.72
VCP P55072 1/20 0.68
MEN1 O00255 3/20 0.61
KMT2A Q03164 3/20 0.61
NPC1 O15118 2/20 0.61
RAB9A P51151 2/20 0.61
POLB P06746 1/20 0.61
NLRP3 Q96P20 1/20 0.61
ALDH1A1 P00352 3/20 0.56
MAPT P10636 2/20 0.56
HSP90AA1 P07900 1/20 0.56
OPRK1 P41145 1/20 0.56
NPSR1 Q6W5P4 1/20 0.56
CES2 O00748 2/20 0.56
CES1 P23141 2/20 0.56
CA1 P00915 1/20 0.52
CA2 P00918 1/20 0.52
HSPD1 P10809 1/20 0.50
TNFRSF1A P19438 1/20 0.50
MAOB P27338 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10069797 0.93 APP (0.72) APPVCPMEN1KMT2ANPC1
SCHEMBL10069794 0.91 APP (0.84) APPVCPMEN1KMT2ANPC1
SCHEMBL10625119 0.86 VCP (0.81) APPVCPMEN1KMT2ANPC1
SCHEMBL27167232 0.85 APP (0.75) APPVCPNPC1RAB9ACES2
SCHEMBL28695966 0.85 APP (0.75) APPVCPNPC1RAB9ACES2
SCHEMBL28629549 0.84 APP (0.73) APPVCPCES2CES1
SCHEMBL10170737 0.84 APP (0.73) APPVCPCES2CES1
SCHEMBL28972824 0.84 APP (0.73) APPVCPMEN1KMT2ANPC1
SCHEMBL28972914 0.84 APP (0.73) APPVCPRAB9AALDH1A1MAPT
SCHEMBL9193189 0.83 FFAR1 (0.60) APPNPC1RAB9APOLBALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 12 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-11691135-B2 Synthesis of alkynones via carbonylative Sonogashira coupling reactions catalyzed by Pd(II)-N-Heterocyclic carbene-pyridine complexes KING FAHD UNIVERSITY OF PETROLEUM & MINERALS (SA) 2023-07-04 US disclosed
CN-115677739-A Preparation method of O, O-boron difluoride complex 华南理工大学 2023-02-03 CN disclosed
US-20220411451-A1 ACTIVE HETEROGENIZED PALLADIUM-BRIDGED-NHC CATALYSTS FOR CARBONYLATIVE SONOGASHIRA COUPLING REACTIONS KING FAHD UNIVERSITY OF PETROLEUM & MINERALS (SA) 2022-12-29 US disclosed
CN-113429280-B Method for preparing chalcone compounds by selective hydrogenation reduction of alkynone under catalysis of Ti (III) complex 陕西师范大学 2022-08-23 CN disclosed
US-20220118435-A1 SYNTHESIS OF ALKYNONES VIA CARBONYLATIVE SONOGASHIRA COUPLING REACTIONS CATALYZED BY PD(II)-N-HETEROCYCLIC CARBENE-PYRIDINE COMPLEXES KING FAHD UNIVERSITY OF PETROLEUM & MINERALS (SA) 2022-04-21 US disclosed
CN-110452270-B Azacarbene palladium complex crystal, synthesis method thereof and application thereof in preparation of alpha, beta-unsaturated ketone compound 陕西师范大学 2022-02-25 CN disclosed
CN-113429280-A Method for preparing chalcone compounds by selective hydrogenation reduction of alkynone under catalysis of Ti (III) complex 陕西师范大学 2021-09-24 CN disclosed
CN-109810147-B Pyrene-labeled benzimidazole nitrogen heterocyclic carbene palladium metal complex, and preparation and application thereof 中国科学院兰州化学物理研究所 2021-02-26 CN disclosed
CN-108148064-B Method for preparing pyrazole quinoxalinone derivative 浙江百斯特化工有限公司 2020-06-26 CN disclosed
CN-101456801-B Method for synthesizing alpha-beta unsaturated acetyenic ketone compounds by carbonylation LANZHOU CHEM PHYS INST 2012-07-04 CN disclosed
WO-2012016619-A1 PHENETHYL, PHENETHYLENE, PHENETHYNE AND INDANONE DERIVATES IN COSMETIC FORMULATIONS, ESPECIALLY FOR USE IN SKIN AGEING PROCESSES MERCK PATENT GMBH (DE) 2012-02-09 WO disclosed
CN-101456801-A Method for synthesizing alpha-beta unsaturated acetyenic ketone compounds by carbonylation LANZHOU CHEM PHYS INST (CN) 2009-06-17 CN disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-11691135-B2 Synthesis of alkynones via carbonylative Sonogashira coupling reactions catalyzed by Pd(II)-N-Heterocyclic carbene-pyridine complexes PDK2, SNCA, YAP1 APP 4235/4885VCP 4072/4885MEN1 1330/4885
US-20220411451-A1 ACTIVE HETEROGENIZED PALLADIUM-BRIDGED-NHC CATALYSTS FOR CARBONYLATIVE SONOGASHIRA COUPLING REACTIONS NDC1, SMARCC2, SMARCC1 APP 4667/4885VCP 3513/4885MEN1 1498/4885
US-20220118435-A1 SYNTHESIS OF ALKYNONES VIA CARBONYLATIVE SONOGASHIRA COUPLING REACTIONS CATALYZED BY PD(II)-N-HETEROCYCLIC CARBENE-PYRIDINE COMPLEXES PDK2, SNCA, YAP1 APP 4235/4885VCP 4072/4885MEN1 1330/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.