SCHEMBL10071172

SCHEMBL10071172

C=C1OB(c2ccc(-c3ccc(NC(=O)OC(C)(C)C)cc3)c(CC)c2)OC1(C)C

nearest known ligand 0.39

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
CYP17A1 P05093 3/20 0.39
PSMB8 P28062 1/20 0.37
CD274 Q9NZQ7 1/20 0.36
HDAC1 Q13547 5/20 0.36
HDAC3 O15379 3/20 0.36
HDAC2 Q92769 2/20 0.36
HDAC8 Q9BY41 2/20 0.36
BRD4 O60885 1/20 0.36
CREBBP Q92793 1/20 0.36
HDAC6 Q9UBN7 4/20 0.35
HDAC10 Q969S8 2/20 0.35
MAP4K4 O95819 1/20 0.35
PRKDC P78527 1/20 0.35
PRMT5 O14744 1/20 0.35
WDR77 Q9BQA1 1/20 0.35
SREBF2 Q12772 1/20 0.35
AAK1 Q2M2I8 1/20 0.34
MAPK14 Q16539 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL402997 0.86 PRMT5 (0.46) CYP17A1PSMB8CD274HDAC1HDAC3
SCHEMBL90904 0.77 AAK1 (0.39) CYP17A1PRMT5WDR77AAK1
SCHEMBL879085 0.75 AAK1 (0.38) PRKDCPRMT5WDR77AAK1
SCHEMBL12316014 0.75 NAMPT (0.39) CYP17A1PSMB8MAP4K4PRMT5WDR77
SCHEMBL408034 0.72 CYP17A1 (0.46) CYP17A1PSMB8CD274HDAC1HDAC3
SCHEMBL12888644 0.71 TSHR (0.36) PSMB8PRMT5WDR77AAK1
SCHEMBL15184583 0.70 AAK1 (0.51) PRMT5WDR77AAK1
SCHEMBL13622824 0.70 SMN1; SMN2 (0.42) BRD4
SCHEMBL1255934 0.70 AAK1 (0.54) CYP17A1PSMB8PRMT5WDR77AAK1
SCHEMBL10382417 0.69 ALDH1A1 (0.51)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20120013245-A1 ELECTROACTIVE MATERIALS E. I. DU PONT DE NEMOURS AND COMPANY (US) 2012-01-19 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20120013245-A1 ELECTROACTIVE MATERIALS NAT1, ADRA1D, ADRA1B CYP17A1 143/4885PSMB8 4174/4885CD274 1302/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.