SCHEMBL10071705

SCHEMBL10071705

O=C(CNC1CCCCC1)c1ccc(O)c(O)c1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.49
HPGD P15428 2/20 0.49
ALPL P05186 3/20 0.49
ALPG P10696 3/20 0.49
MEN1 O00255 2/20 0.47
KMT2A Q03164 2/20 0.47
SLC2A1 P11166 1/20 0.46
CXCR4 P61073 1/20 0.46
PABPC1 P11940 1/20 0.45
ERCC1 P07992 2/20 0.45
ERCC4 Q92889 2/20 0.45
HDAC1 Q13547 2/20 0.44
HDAC6 Q9UBN7 1/20 0.41
PLAA Q9Y263 2/20 0.41
KDM4E B2RXH2 2/20 0.41
GAA P10253 2/20 0.41
MAPT P10636 2/20 0.41
CA12 O43570 1/20 0.41
CA1 P00915 1/20 0.41
CA2 P00918 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9768072 0.98 ALPG (0.48) ALDH1A1HPGDALPLALPGMEN1
SCHEMBL6890171 0.78 MEN1 (0.62) ALDH1A1HPGDMEN1KMT2AKDM4E
SCHEMBL19144755 0.76 MEN1 (0.45) ALDH1A1HPGDMEN1KMT2ACXCR4
SCHEMBL8930279 0.76 MEN1 (0.60) ALDH1A1HPGDMEN1KMT2AKDM4E
SCHEMBL9768145 0.75 ALPG (0.46) ALPLALPGERCC1ERCC4HDAC1
SCHEMBL5325765 0.73 ALDH1A1 (0.49) ALDH1A1HPGDMEN1KMT2ACXCR4
Adrenalone SCHEMBL29550997 0.72 ALPG (0.55) ALPLALPGMEN1KMT2AHDAC6
SCHEMBL14646958 0.72 ALPG (0.51) ALPLALPGHDAC6PLAAKDM4E
Adrenalone SCHEMBL123124 0.72 ALPG (0.55) ALPLALPGMEN1KMT2AHDAC6
SCHEMBL9768178 0.71 KDM4E (0.53) ALDH1A1HPGDALPLALPGMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9266817-B2 Catecholamine derivatives for obesity and neurological disorders EMORY UNIVERSITY (US) 2016-02-23 US disclosed
US-20140329907-A1 CATECHOLAMINE DERIVATIVES FOR OBESITY AND NEUROLOGICAL DISORDERS NATIONAL INSTITUTES OF HEALTH (NIH), U.S. DEPT. OF HEALTH AND HUMAN SERVICES (DHHS), U.S. GOVERNMENT 2014-11-06 US disclosed
US-20120022086-A1 CATECHOLAMINE DERIVATIVES FOR OBESITY AND NEUROLOGICAL DISORDERS EMORY UNIVERSITY (US) 2012-01-26 US disclosed
WO-2010107866-A2 CATECHOLAMINE DERIVATIVES FOR OBESITY AND NEUROLOGICAL DISORDERS EMORY UNIVERSITY (US) 2010-09-23 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20120022086-A1 CATECHOLAMINE DERIVATIVES FOR OBESITY AND NEUROLOGICAL DISORDERS BDNF, NTRK2, COMT ALDH1A1 412/4885HPGD 1609/4885ALPL 4539/4885
US-20140329907-A1 CATECHOLAMINE DERIVATIVES FOR OBESITY AND NEUROLOGICAL DISORDERS BDNF, NTRK2, COMT ALDH1A1 412/4885HPGD 1609/4885ALPL 4539/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.