Dimethylaminoethanol

Dimethylaminoethanol

SCHEMBL1007646

Br.CN(C)CCO.CN(C)CCO.Cl

nearest known ligand 0.86

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

ACHEADRA1AADRA1BADRA1DADRA2AADRA2BADRA2CADRB1ADRB2ADRB3APH1AAPH1BCHRM2CHRM3EZH2GRIN2AHTR1AHTR1BHTR1DHTR1FHTR3ANCSTNP2RY12PSEN1PSEN2PSENENSIGMAR1SLC6A2SLC6A3SLC6A4

The experimentally established mechanism targets of Dimethylaminoethanol. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CHRM2 known ✓ P08172 1/20 0.31
CHRM3 known ✓ P20309 1/20 0.31
MAPT P10636 1/20 0.86
ALDH1A1 P00352 2/20 0.39
TDP1 Q9NUW8 2/20 0.39
CA12 O43570 2/20 0.39
CA2 P00918 2/20 0.39
CA9 Q16790 2/20 0.39
TSHR P16473 1/20 0.39
CA3 P07451 1/20 0.39
CA4 P22748 1/20 0.39
CA6 P23280 1/20 0.39
CA5A P35218 1/20 0.39
CA7 P43166 1/20 0.39
CA14 Q9ULX7 1/20 0.39
CA5B Q9Y2D0 1/20 0.39
DNM1 Q05193 3/20 0.36
PRMT3 O60678 1/20 0.33
CARM1 Q86X55 1/20 0.33
PRMT6 Q96LA8 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 56 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020065541-A1 MICROEMULSIONS AND METHODS OF USE MOROCCANOIL ISRAEL, LTD. (IL) 2020-04-02 WO claimed
CN-104884198-B The method for preparing the hollow metal nanometer particle being supported on carrier LG化学株式会社 2017-11-17 CN claimed
US-20120003319-A9 COMPOSITIONS FOR SITE-SPECIFIC DELIVERY OF IMATINIB AND METHODS OF USE ELAN PHARMA INTERNATIONAL LIMITED (IE) 2012-01-05 US claimed
EP-2271316-A2 FENOFIBRATE DOSAGE FORMS Elan Pharma International Limited (IE) 2011-01-12 EP claimed
EP-2268265-A2 COMPOSITIONS FOR SITE-SPECIFIC DELIVERY OF IMATINIB AND METHODS OF USE Elan Pharma International Limited (IE) 2011-01-05 EP claimed
US-7842232-B2 Sterilization of dispersions of nanoparticulate active agents with gamma radiation ELAN PHARMA INTERNATIONAL, LTD. (IE) 2010-11-30 US claimed
US-20090269400-A1 Nanoparticulate and Controlled Release Compositions Comprising a Cephalosporin ELAN PHARMA INTERNATIONAL LIMITED (IE) 2009-10-29 US claimed
WO-2009120919-A2 FENOFIBRATE DOSAGE FORMS ELAN PHARMA INTERNATIONAL LTD. (IE) 2009-10-01 WO claimed
WO-2009117401-A2 COMPOSITIONS FOR SITE-SPECIFIC DELIVERY OF IMATINIB AND METHODS OF USE ELAN PHARAMA INTERNATIONAL LIMITED (IE) 2009-09-24 WO claimed
US-20090238884-A1 COMPOSITIONS FOR SITE-SPECIFIC DELIVERY OF IMATINIB AND METHODS OF USE ELAN PHARMA INTERNATIONAL LIMITED (IE) 2009-09-24 US claimed
EP-1855651-A1 NANOPARTICULATE COMPOSITIONS OF HETEROCYCLIC AMIDE DERIVATIVES Elan Pharma International Limited (IE) 2007-11-21 EP claimed
WO-2007100466-A2 NANOPARTICULATE CARVEDILOL FORMULATIONS ELAN PHARMA INTERNATIONAL LTD. (IE) 2007-09-07 WO claimed
EP-1809279-A1 NANOPARTICULATE COMPOSITIONS OF TUBULIN INHIBITOR BAXTER INTERNATIONAL INC. (US) 2007-07-25 EP claimed
US-20060210638-A1 Injectable compositions of nanoparticulate immunosuppressive compounds ELAN PHARMA INTERNATIONAL LIMITED 2006-09-21 US claimed
WO-2006096462-A1 NANOPARTICULATE COMPOSITIONS OF HETEROCYCLIC AMIDE DERIVATIVES ELAN PHARMA INTERNATIONAL LIMITED (IE) 2006-09-14 WO claimed
WO-2006052712-A1 NANOPARTICULATE COMPOSITIONS OF TUBULIN INHIBITOR BAXTER INTERNATIONAL INC. (US) 2006-05-18 WO claimed
US-20050233001-A1 Nanoparticulate megestrol formulations ELAN PHARMA INTERNATIONAL LTD. 2005-10-20 US claimed
US-20050004049-A1 Novel griseofulvin compositions ELAN PHARMA INTERNATIONAL LIMITED 2005-01-06 US claimed
US-20040033202-A1 Nanoparticulate sterol formulations and novel sterol combinations ELAN PHARMA INTERNATIONAL, LTD. 2004-02-19 US claimed
US-20030224058-A1 Fibrate particles of an effective average particle size of less than 2000 nm. having a stabilizer associated with the surface; improved pharmacokinetic profiles and reduced fed/fasted variability. ELAN PHARMA INTERNATIONAL, LTD. 2003-12-04 US claimed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (5 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20060210638-A1 Injectable compositions of nanoparticulate immunosuppressive compounds RPTOR, IMMT, FKBP4 CHRM2 4259/4885CHRM3 3914/4885MAPT 1103/4885
US-20090238884-A1 COMPOSITIONS FOR SITE-SPECIFIC DELIVERY OF IMATINIB AND METHODS OF USE ABL1, SI, ABL2 CHRM2 2748/4885CHRM3 1557/4885MAPT 2929/4885
US-20090269400-A1 Nanoparticulate and Controlled Release Compositions Comprising a Cephalosporin CLSPN, ABCB11, SLC47A1 CHRM2 1459/4885CHRM3 2460/4885MAPT 3209/4885
US-20120003319-A9 COMPOSITIONS FOR SITE-SPECIFIC DELIVERY OF IMATINIB AND METHODS OF USE ABL1, SI, ABL2 CHRM2 2748/4885CHRM3 1557/4885MAPT 2929/4885
US-20050004049-A1 Novel griseofulvin compositions GRN, GRM5, GRM3 CHRM2 1630/4885CHRM3 1483/4885MAPT 1538/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.