SCHEMBL10083992

SCHEMBL10083992

O=C(NC(CN1CCCC1)c1ccccc1)C1(c2cccnc2)CC1

nearest known ligand 0.44

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ITGA4 P13612 6/20 0.44
ITGB7 P26010 6/20 0.44
ROCK2 O75116 2/20 0.41
ROCK1 Q13464 2/20 0.41
PIN1 Q13526 1/20 0.41
MEN1 O00255 1/20 0.40
KMT2A Q03164 1/20 0.40
ALDH1A1 P00352 1/20 0.40
LMNA P02545 1/20 0.40
OPRM1 P35372 1/20 0.40
OPRD1 P41143 1/20 0.40
OPRK1 P41145 1/20 0.40
OPRL1 P41146 1/20 0.40
HSD11B1 P28845 2/20 0.40
GPR88 Q9GZN0 1/20 0.39
AURKA O14965 1/20 0.39
RPS6KB1 P23443 1/20 0.39
AURKB Q96GD4 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15385500 1.00 ITGA4 (0.44) ITGA4ITGB7ROCK2ROCK1PIN1
Hydrochloric Acid SCHEMBL432371 0.99 ITGA4 (0.44) ITGA4ITGB7ROCK2ROCK1PIN1
Hydrochloric Acid SCHEMBL432370 0.99 ITGA4 (0.44) ITGA4ITGB7ROCK2ROCK1PIN1
SCHEMBL15385492 0.89 HSD11B1 (0.50) MEN1KMT2AALDH1A1HSD11B1GPR88
SCHEMBL435831 0.89 HSD11B1 (0.50) MEN1KMT2AALDH1A1HSD11B1GPR88
SCHEMBL433057 0.88 ROCK2 (0.48) ITGA4ITGB7ROCK2ROCK1KMT2A
SCHEMBL433056 0.88 ROCK2 (0.48) ITGA4ITGB7ROCK2ROCK1KMT2A
Hydrochloric Acid SCHEMBL434246 0.88 HSD11B1 (0.49) MEN1KMT2AALDH1A1OPRM1OPRD1
Hydrochloric Acid SCHEMBL15380695 0.88 HSD11B1 (0.49) MEN1KMT2AALDH1A1OPRM1OPRD1
SCHEMBL10083337 0.84 MEN1 (0.52) MEN1KMT2AALDH1A1LMNAHSD11B1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012012410-A2 KAPPA OPIOID RECEPTOR AGONISTS DR. REDDY'S LABORATORIES LTD. (IN) 2012-01-26 WO disclosed