SCHEMBL100906

SCHEMBL100906

O=C(O)Nc1cc(CCC(=O)Nc2ccc3sc(CO)cc3c2)ccc1-c1ccccc1

nearest known ligand 0.42

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
HDAC1 Q13547 2/20 0.42
AKR1C3 P42330 1/20 0.41
AKR1C2 P52895 1/20 0.41
MAPT P10636 6/20 0.40
GAA P10253 1/20 0.40
HCAR2 Q8TDS4 3/20 0.40
PLAU P00749 1/20 0.39
RAB9A P51151 3/20 0.39
NPC1 O15118 2/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
LMNA P02545 1/20 0.39
TP53 P04637 1/20 0.39
POLB P06746 1/20 0.39
TOP2A P11388 1/20 0.38
TOP2B Q02880 1/20 0.38
HTT P42858 1/20 0.38
RORC P51449 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL99215 0.84 AKR1C3 (0.49) HDAC1AKR1C3AKR1C2MAPTGAA
SCHEMBL661537 0.82 CHRM3 (0.51)
SCHEMBL98704 0.82 AKR1C3 (0.51) HDAC1AKR1C3AKR1C2MAPTGAA
Iodide SCHEMBL99557 0.82 CHRM3 (0.37) HDAC1
SCHEMBL101249 0.80 AKR1C3 (0.45) AKR1C3AKR1C2MAPTGAAHCAR2
SCHEMBL100326 0.79 HCAR2 (0.46) HDAC1AKR1C3AKR1C2MAPTGAA
SCHEMBL100587 0.78 RORC (0.46) HDAC1AKR1C3AKR1C2MAPTGAA
SCHEMBL100288 0.78 PTGDR2 (0.46) HDAC1AKR1C3AKR1C2MAPTGAA
SCHEMBL99412 0.78 HCAR2 (0.47) HDAC1AKR1C3AKR1C2MAPTHCAR2
SCHEMBL15821963 0.77 AKR1C3 (0.50) HDAC1AKR1C3AKR1C2MAPTGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2426121-A1 QUATERNARY AMMONIUM SALT COMPOUND Teijin Pharma Limited (JP) 2012-03-07 EP claimed