SCHEMBL1009811

SCHEMBL1009811

c1ccc(N[N]c2cc[nH]n2)cc1

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TDP1 Q9NUW8 4/20 0.35
TSHR P16473 3/20 0.35
CYP1A1 P04798 1/20 0.35
CYP1B1 Q16678 1/20 0.35
NOX1 Q9Y5S8 1/20 0.34
DEPTOR Q8TB45 1/20 0.33
MAPT P10636 8/20 0.32
GAA P10253 7/20 0.32
ALDH1A1 P00352 6/20 0.32
MEN1 O00255 5/20 0.32
KMT2A Q03164 5/20 0.32
TAAR1 Q96RJ0 2/20 0.32
KDM4E B2RXH2 1/20 0.32
HPGD P15428 4/20 0.32
RAB9A P51151 3/20 0.32
NPC1 O15118 2/20 0.32
SMN1; SMN2 Q16637 1/20 0.32
LMNA P02545 3/20 0.32
HSD17B10 Q99714 3/20 0.31
CTSD P07339 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2108118 0.81 CYP1A1 (0.50) TDP1TSHRCYP1A1CYP1B1NOX1
Benzene SCHEMBL11416188 0.72 MAOA (0.32)
SCHEMBL9349266 0.68 MAPT (0.39) MAPTALDH1A1TAAR1L3MBTL1
SCHEMBL5560073 0.68 ADRA2A (0.50) TDP1TSHRCYP1A1CYP1B1NOX1
SCHEMBL3064895 0.68 ALDH1A1 (0.50) TDP1TSHRMAPTGAAALDH1A1
SCHEMBL2554754 0.68 ALDH1A1 (0.50) TDP1TSHRMAPTGAAALDH1A1
Azobenzene SCHEMBL11590710 0.68 ALDH1A1 (0.50) TDP1TSHRMAPTGAAALDH1A1
SCHEMBL1569120 0.68
SCHEMBL5754707 0.67 MAPT (0.48) TDP1MAPTGAAALDH1A1MEN1
SCHEMBL5751505 0.67 MAPT (0.48) TDP1MAPTGAAALDH1A1MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1824489-B1 STEREOISOMERICALLY ENRICHED 3-AMINOCARBONYL BICYCLOHEPTENE PYRIMIDINEDIAMINE COMPOUNDS AND THEIR USES RIGEL PHARMACEUTICALS INC (US) 2011-01-05 EP disclosed